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A Cereblon Modulator (CC-220) with Improved Degradation of Ikaros and Aiolos.
Matyskiela, Mary E; Zhang, Weihong; Man, Hon-Wah; Muller, George; Khambatta, Godrej; Baculi, Frans; Hickman, Matthew; LeBrun, Laurie; Pagarigan, Barbra; Carmel, Gilles; Lu, Chin-Chun; Lu, Gang; Riley, Mariko; Satoh, Yoshitaka; Schafer, Peter; Daniel, Thomas O; Carmichael, James; Cathers, Brian E; Chamberlain, Philip P.
Affiliation
  • Matyskiela ME; 1Celgene Corporation , 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Zhang W; 1Celgene Corporation , 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Man HW; 1Celgene Corporation , 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Muller G; 1Celgene Corporation , 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Khambatta G; 1Celgene Corporation , 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Baculi F; 1Celgene Corporation , 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Hickman M; 1Celgene Corporation , 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • LeBrun L; 1Celgene Corporation , 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Pagarigan B; 1Celgene Corporation , 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Carmel G; 1Celgene Corporation , 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Lu CC; 1Celgene Corporation , 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Lu G; 1Celgene Corporation , 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Riley M; 1Celgene Corporation , 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Satoh Y; 1Celgene Corporation , 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Schafer P; 1Celgene Corporation , 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Daniel TO; 1Celgene Corporation , 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Carmichael J; 1Celgene Corporation , 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Cathers BE; 1Celgene Corporation , 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
  • Chamberlain PP; 1Celgene Corporation , 10300 Campus Point Drive, Suite 100, San Diego, California 92121, United States.
J Med Chem ; 61(2): 535-542, 2018 01 25.
Article in En | MEDLINE | ID: mdl-28425720

Full text: 1 Database: MEDLINE Main subject: Peptide Hydrolases / Ikaros Transcription Factor / Proteolysis / Heterocyclic Compounds, 4 or More Rings Type of study: Prognostic_studies Limits: Humans Language: En Journal: J Med Chem Journal subject: QUIMICA Year: 2018 Type: Article Affiliation country: United States

Full text: 1 Database: MEDLINE Main subject: Peptide Hydrolases / Ikaros Transcription Factor / Proteolysis / Heterocyclic Compounds, 4 or More Rings Type of study: Prognostic_studies Limits: Humans Language: En Journal: J Med Chem Journal subject: QUIMICA Year: 2018 Type: Article Affiliation country: United States