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Crystal structures of agonist-bound human cannabinoid receptor CB1.
Hua, Tian; Vemuri, Kiran; Nikas, Spyros P; Laprairie, Robert B; Wu, Yiran; Qu, Lu; Pu, Mengchen; Korde, Anisha; Jiang, Shan; Ho, Jo-Hao; Han, Gye Won; Ding, Kang; Li, Xuanxuan; Liu, Haiguang; Hanson, Michael A; Zhao, Suwen; Bohn, Laura M; Makriyannis, Alexandros; Stevens, Raymond C; Liu, Zhi-Jie.
Affiliation
  • Hua T; iHuman Institute, ShanghaiTech University, Shanghai 201210, China.
  • Vemuri K; National Laboratory of Biomacromolecules, Institute of Biophysics, Chinese Academy of Sciences, Beijing 100101, China.
  • Nikas SP; University of Chinese Academy of Sciences, Beijing 100049, China.
  • Laprairie RB; Center for Drug Discovery, Department of Pharmaceutical Sciences; Department of Chemistry and Chemical Biology, Northeastern University, Boston, Massachusetts 02115, USA.
  • Wu Y; Center for Drug Discovery, Department of Pharmaceutical Sciences; Department of Chemistry and Chemical Biology, Northeastern University, Boston, Massachusetts 02115, USA.
  • Qu L; Departments of Molecular Medicine and Neuroscience, The Scripps Research Institute, Jupiter, Florida 33458, USA.
  • Pu M; iHuman Institute, ShanghaiTech University, Shanghai 201210, China.
  • Korde A; iHuman Institute, ShanghaiTech University, Shanghai 201210, China.
  • Jiang S; National Laboratory of Biomacromolecules, Institute of Biophysics, Chinese Academy of Sciences, Beijing 100101, China.
  • Ho JH; University of Chinese Academy of Sciences, Beijing 100049, China.
  • Han GW; iHuman Institute, ShanghaiTech University, Shanghai 201210, China.
  • Ding K; Center for Drug Discovery, Department of Pharmaceutical Sciences; Department of Chemistry and Chemical Biology, Northeastern University, Boston, Massachusetts 02115, USA.
  • Li X; Center for Drug Discovery, Department of Pharmaceutical Sciences; Department of Chemistry and Chemical Biology, Northeastern University, Boston, Massachusetts 02115, USA.
  • Liu H; Departments of Molecular Medicine and Neuroscience, The Scripps Research Institute, Jupiter, Florida 33458, USA.
  • Hanson MA; Departments of Biological Sciences and Chemistry, Bridge Institute, University of Southern California, Los Angeles, California 90089, USA.
  • Zhao S; iHuman Institute, ShanghaiTech University, Shanghai 201210, China.
  • Bohn LM; University of Chinese Academy of Sciences, Beijing 100049, China.
  • Makriyannis A; School of Life Science and Technology, ShanghaiTech University, Shanghai 201210, China.
  • Stevens RC; Complex Systems Division, Beijing Computational Science Research Center, Beijing 100193, China.
  • Liu ZJ; Complex Systems Division, Beijing Computational Science Research Center, Beijing 100193, China.
Nature ; 547(7664): 468-471, 2017 07 27.
Article in En | MEDLINE | ID: mdl-28678776

Full text: 1 Database: MEDLINE Main subject: Dronabinol / Receptor, Cannabinoid, CB1 / Droperidol / Cannabinoid Receptor Agonists Type of study: Prognostic_studies Limits: Humans Language: En Journal: Nature Year: 2017 Type: Article Affiliation country: China

Full text: 1 Database: MEDLINE Main subject: Dronabinol / Receptor, Cannabinoid, CB1 / Droperidol / Cannabinoid Receptor Agonists Type of study: Prognostic_studies Limits: Humans Language: En Journal: Nature Year: 2017 Type: Article Affiliation country: China