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Allosteric Inhibitors, Crystallography, and Comparative Analysis Reveal Network of Coordinated Movement across Human Herpesvirus Proteases.
Acker, Timothy M; Gable, Jonathan E; Bohn, Markus-Frederik; Jaishankar, Priyadarshini; Thompson, Michael C; Fraser, James S; Renslo, Adam R; Craik, Charles S.
Affiliation
  • Acker TM; Department of Pharmaceutical Chemistry, University of California , San Francisco, California 94158, United States.
  • Gable JE; Department of Pharmaceutical Chemistry, University of California , San Francisco, California 94158, United States.
  • Bohn MF; Department of Pharmaceutical Chemistry, University of California , San Francisco, California 94158, United States.
  • Jaishankar P; Department of Pharmaceutical Chemistry, University of California , San Francisco, California 94158, United States.
  • Thompson MC; Department of Bioengineering and Therapeutic Sciences, University of California , San Francisco, California 94158, United States.
  • Fraser JS; Department of Bioengineering and Therapeutic Sciences, University of California , San Francisco, California 94158, United States.
  • Renslo AR; Department of Pharmaceutical Chemistry, University of California , San Francisco, California 94158, United States.
  • Craik CS; Department of Pharmaceutical Chemistry, University of California , San Francisco, California 94158, United States.
J Am Chem Soc ; 139(34): 11650-11653, 2017 08 30.
Article in En | MEDLINE | ID: mdl-28759216

Full text: 1 Database: MEDLINE Main subject: Peptide Hydrolases / Protease Inhibitors / Herpesviridae Infections / Herpesvirus 8, Human / Allosteric Regulation Limits: Humans Language: En Journal: J Am Chem Soc Year: 2017 Type: Article Affiliation country: United States

Full text: 1 Database: MEDLINE Main subject: Peptide Hydrolases / Protease Inhibitors / Herpesviridae Infections / Herpesvirus 8, Human / Allosteric Regulation Limits: Humans Language: En Journal: J Am Chem Soc Year: 2017 Type: Article Affiliation country: United States