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Targeting STING with covalent small-molecule inhibitors.
Haag, Simone M; Gulen, Muhammet F; Reymond, Luc; Gibelin, Antoine; Abrami, Laurence; Decout, Alexiane; Heymann, Michael; van der Goot, F Gisou; Turcatti, Gerardo; Behrendt, Rayk; Ablasser, Andrea.
Affiliation
  • Haag SM; Global Health Institute, Swiss Federal Institute of Technology Lausanne (EPFL), Lausanne, Switzerland.
  • Gulen MF; Global Health Institute, Swiss Federal Institute of Technology Lausanne (EPFL), Lausanne, Switzerland.
  • Reymond L; Biomolecular Screening Facility, Swiss Federal Institute of Technology Lausanne (EPFL), Lausanne, Switzerland.
  • Gibelin A; Biomolecular Screening Facility, Swiss Federal Institute of Technology Lausanne (EPFL), Lausanne, Switzerland.
  • Abrami L; Global Health Institute, Swiss Federal Institute of Technology Lausanne (EPFL), Lausanne, Switzerland.
  • Decout A; Global Health Institute, Swiss Federal Institute of Technology Lausanne (EPFL), Lausanne, Switzerland.
  • Heymann M; Global Health Institute, Swiss Federal Institute of Technology Lausanne (EPFL), Lausanne, Switzerland.
  • van der Goot FG; Global Health Institute, Swiss Federal Institute of Technology Lausanne (EPFL), Lausanne, Switzerland.
  • Turcatti G; Biomolecular Screening Facility, Swiss Federal Institute of Technology Lausanne (EPFL), Lausanne, Switzerland.
  • Behrendt R; Institute for Immunology, Faculty of Medicine, Technical University Dresden, Dresden, Germany.
  • Ablasser A; Global Health Institute, Swiss Federal Institute of Technology Lausanne (EPFL), Lausanne, Switzerland. andrea.ablasser@epfl.ch.
Nature ; 559(7713): 269-273, 2018 07.
Article in En | MEDLINE | ID: mdl-29973723

Full text: 1 Database: MEDLINE Main subject: Small Molecule Libraries / Membrane Proteins Type of study: Prognostic_studies Limits: Animals / Humans Language: En Journal: Nature Year: 2018 Type: Article Affiliation country: Switzerland

Full text: 1 Database: MEDLINE Main subject: Small Molecule Libraries / Membrane Proteins Type of study: Prognostic_studies Limits: Animals / Humans Language: En Journal: Nature Year: 2018 Type: Article Affiliation country: Switzerland