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Synthesis and evaluation of tetrahydropyrazolopyridine inhibitors of anion exchange protein SLC26A4 (pendrin).
Zhu, Jie S; Lu, Julia Y; Tan, Joseph-Anthony; Rivera, Amber A; Phuan, Puay-Wah; Shatskikh, Marina E; Son, Jung-Ho; Haggie, Peter M; Verkman, Alan S; Kurth, Mark J.
Affiliation
  • Zhu JS; Department of Chemistry, University of California, Davis, CA 95616, United States.
  • Lu JY; Department of Chemistry, University of California, Davis, CA 95616, United States.
  • Tan JA; Departments of Medicine & Physiology, University of California, San Francisco, CA 94143, United States.
  • Rivera AA; Departments of Medicine & Physiology, University of California, San Francisco, CA 94143, United States.
  • Phuan PW; Departments of Medicine & Physiology, University of California, San Francisco, CA 94143, United States.
  • Shatskikh ME; Department of Chemistry, University of California, Davis, CA 95616, United States.
  • Son JH; Department of Chemistry, University of California, Davis, CA 95616, United States.
  • Haggie PM; Departments of Medicine & Physiology, University of California, San Francisco, CA 94143, United States.
  • Verkman AS; Departments of Medicine & Physiology, University of California, San Francisco, CA 94143, United States.
  • Kurth MJ; Department of Chemistry, University of California, Davis, CA 95616, United States. Electronic address: mjkurth@ucdavis.edu.
Bioorg Med Chem Lett ; 29(16): 2119-2123, 2019 08 15.
Article in En | MEDLINE | ID: mdl-31281021

Full text: 1 Database: MEDLINE Main subject: Pyrazoles / Pyridines / Sulfate Transporters Limits: Animals Language: En Journal: Bioorg Med Chem Lett Journal subject: BIOQUIMICA / QUIMICA Year: 2019 Type: Article Affiliation country: United States

Full text: 1 Database: MEDLINE Main subject: Pyrazoles / Pyridines / Sulfate Transporters Limits: Animals Language: En Journal: Bioorg Med Chem Lett Journal subject: BIOQUIMICA / QUIMICA Year: 2019 Type: Article Affiliation country: United States