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Clinically Relevant OATP2B1 Inhibitors in Marketed Drug Space.
Unger, Melissa S; Mudunuru, Jennypher; Schwab, Matthias; Hopf, Carsten; Drewes, Gerard; Nies, Anne T; Zamek-Gliszczynski, Maciej J; Reinhard, Friedrich B M.
Affiliation
  • Unger MS; Cellzome, a GlaxoSmithKline Company , 69117 Heidelberg , Germany.
  • Mudunuru J; Center for Mass Spectrometry and Optical Spectroscopy (CeMOS) and Institute of Medical Technology , Heidelberg University and Mannheim University of Applied Sciences , 68163 Mannheim , Germany.
  • Schwab M; Drug Metabolism and Disposition , GlaxoSmithKline , Collegeville , Pennsylvania 19426 , United States.
  • Hopf C; Dr. Margarete Fischer-Bosch Institute of Clinical Pharmacology , University of Tübingen , 70376 Stuttgart , Germany.
  • Drewes G; Departments of Clinical Pharmacology, Pharmacy and Biochemistry , University of Tübingen , 72074 Tübingen , Germany.
  • Nies AT; Center for Mass Spectrometry and Optical Spectroscopy (CeMOS) and Institute of Medical Technology , Heidelberg University and Mannheim University of Applied Sciences , 68163 Mannheim , Germany.
  • Zamek-Gliszczynski MJ; Cellzome, a GlaxoSmithKline Company , 69117 Heidelberg , Germany.
  • Reinhard FBM; Dr. Margarete Fischer-Bosch Institute of Clinical Pharmacology , University of Tübingen , 70376 Stuttgart , Germany.
Mol Pharm ; 17(2): 488-498, 2020 02 03.
Article in En | MEDLINE | ID: mdl-31834804

Full text: 1 Database: MEDLINE Main subject: Organic Anion Transporters / Drug Evaluation, Preclinical Type of study: Guideline / Risk_factors_studies Limits: Humans Language: En Journal: Mol Pharm Journal subject: BIOLOGIA MOLECULAR / FARMACIA / FARMACOLOGIA Year: 2020 Type: Article Affiliation country: Germany

Full text: 1 Database: MEDLINE Main subject: Organic Anion Transporters / Drug Evaluation, Preclinical Type of study: Guideline / Risk_factors_studies Limits: Humans Language: En Journal: Mol Pharm Journal subject: BIOLOGIA MOLECULAR / FARMACIA / FARMACOLOGIA Year: 2020 Type: Article Affiliation country: Germany