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Synthesis and evaluation of sulfonyl piperazine LpxH inhibitors.
Kwak, Seung-Hwa; Cochrane, C Skyler; Ennis, Amanda F; Lim, Won Young; Webster, Caroline G; Cho, Jae; Fenton, Benjamin A; Zhou, Pei; Hong, Jiyong.
Affiliation
  • Kwak SH; Department of Chemistry, Duke University, Durham, NC 27708, United States.
  • Cochrane CS; Department of Chemistry, Duke University, Durham, NC 27708, United States.
  • Ennis AF; Department of Chemistry, Duke University, Durham, NC 27708, United States.
  • Lim WY; Department of Chemistry, Duke University, Durham, NC 27708, United States.
  • Webster CG; Department of Chemistry, Duke University, Durham, NC 27708, United States.
  • Cho J; Department of Biochemistry, Duke University Medical Center, Durham, NC 27710, United States.
  • Fenton BA; Department of Biochemistry, Duke University Medical Center, Durham, NC 27710, United States.
  • Zhou P; Department of Chemistry, Duke University, Durham, NC 27708, United States; Department of Biochemistry, Duke University Medical Center, Durham, NC 27710, United States. Electronic address: peizhou@biochem.duke.edu.
  • Hong J; Department of Chemistry, Duke University, Durham, NC 27708, United States; Department of Pharmacology and Cancer Biology, Duke University Medical Center, Durham, NC, 27710, United States. Electronic address: jiyong.hong@duke.edu.
Bioorg Chem ; 102: 104055, 2020 09.
Article in En | MEDLINE | ID: mdl-32663666

Full text: 1 Database: MEDLINE Main subject: Enzyme Inhibitors / Piperazine / Antinematodal Agents Limits: Humans Language: En Journal: Bioorg Chem Year: 2020 Type: Article Affiliation country: United States

Full text: 1 Database: MEDLINE Main subject: Enzyme Inhibitors / Piperazine / Antinematodal Agents Limits: Humans Language: En Journal: Bioorg Chem Year: 2020 Type: Article Affiliation country: United States