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Identification of unprecedented ATP-competitive choline kinase inhibitors.
Quartieri, Francesca; Nesi, Marcella; Avanzi, Nilla R; Borghi, Daniela; Casale, Elena; Corti, Emiliana; Cucchi, Ulisse; Donati, Daniele; Fasolini, Marina; Felder, Eduard R; Galvani, Arturo; Giorgini, Maria L; Lomolino, Antonio; Menichincheri, Maria; Orrenius, Christian; Perrera, Claudia; Re Depaolini, Stefania; Riccardi-Sirtori, Federico; Salsi, Enea; Isacchi, Antonella; Gnocchi, Paola.
Affiliation
  • Quartieri F; Nerviano Medical Sciences Srl, Viale Pasteur 10, 20014 Nerviano (MI), Italy. Electronic address: francesca.quartieri@nervianoms.com.
  • Nesi M; Nerviano Medical Sciences Srl, Viale Pasteur 10, 20014 Nerviano (MI), Italy.
  • Avanzi NR; Nerviano Medical Sciences Srl, Viale Pasteur 10, 20014 Nerviano (MI), Italy.
  • Borghi D; Nerviano Medical Sciences Srl, Viale Pasteur 10, 20014 Nerviano (MI), Italy.
  • Casale E; Nerviano Medical Sciences Srl, Viale Pasteur 10, 20014 Nerviano (MI), Italy.
  • Corti E; Nerviano Medical Sciences Srl, Viale Pasteur 10, 20014 Nerviano (MI), Italy.
  • Cucchi U; Nerviano Medical Sciences Srl, Viale Pasteur 10, 20014 Nerviano (MI), Italy.
  • Donati D; Nerviano Medical Sciences Srl, Viale Pasteur 10, 20014 Nerviano (MI), Italy.
  • Fasolini M; Nerviano Medical Sciences Srl, Viale Pasteur 10, 20014 Nerviano (MI), Italy.
  • Felder ER; Nerviano Medical Sciences Srl, Viale Pasteur 10, 20014 Nerviano (MI), Italy.
  • Galvani A; Nerviano Medical Sciences Srl, Viale Pasteur 10, 20014 Nerviano (MI), Italy.
  • Giorgini ML; Nerviano Medical Sciences Srl, Viale Pasteur 10, 20014 Nerviano (MI), Italy.
  • Lomolino A; Nerviano Medical Sciences Srl, Viale Pasteur 10, 20014 Nerviano (MI), Italy.
  • Menichincheri M; Nerviano Medical Sciences Srl, Viale Pasteur 10, 20014 Nerviano (MI), Italy.
  • Orrenius C; Nerviano Medical Sciences Srl, Viale Pasteur 10, 20014 Nerviano (MI), Italy.
  • Perrera C; Nerviano Medical Sciences Srl, Viale Pasteur 10, 20014 Nerviano (MI), Italy.
  • Re Depaolini S; Nerviano Medical Sciences Srl, Viale Pasteur 10, 20014 Nerviano (MI), Italy.
  • Riccardi-Sirtori F; Nerviano Medical Sciences Srl, Viale Pasteur 10, 20014 Nerviano (MI), Italy.
  • Salsi E; Nerviano Medical Sciences Srl, Viale Pasteur 10, 20014 Nerviano (MI), Italy.
  • Isacchi A; Nerviano Medical Sciences Srl, Viale Pasteur 10, 20014 Nerviano (MI), Italy.
  • Gnocchi P; Nerviano Medical Sciences Srl, Viale Pasteur 10, 20014 Nerviano (MI), Italy.
Bioorg Med Chem Lett ; 51: 128310, 2021 11 01.
Article in En | MEDLINE | ID: mdl-34416377

Full text: 1 Database: MEDLINE Main subject: Adenosine Triphosphate / Choline Kinase / Cyclohexanes / Protein Kinase Inhibitors Type of study: Diagnostic_studies Limits: Humans Language: En Journal: Bioorg Med Chem Lett Journal subject: BIOQUIMICA / QUIMICA Year: 2021 Type: Article

Full text: 1 Database: MEDLINE Main subject: Adenosine Triphosphate / Choline Kinase / Cyclohexanes / Protein Kinase Inhibitors Type of study: Diagnostic_studies Limits: Humans Language: En Journal: Bioorg Med Chem Lett Journal subject: BIOQUIMICA / QUIMICA Year: 2021 Type: Article