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The Interleukin-1 Receptor-Associated Kinase 4 Inhibitor PF-06650833 Blocks Inflammation in Preclinical Models of Rheumatic Disease and in Humans Enrolled in a Randomized Clinical Trial.
Winkler, Aaron; Sun, Weiyong; De, Saurav; Jiao, Aiping; Sharif, M Nusrat; Symanowicz, Peter T; Athale, Shruti; Shin, Julia H; Wang, Ju; Jacobson, Bruce A; Ramsey, Simeon J; Dower, Ken; Andreyeva, Tatyana; Liu, Heng; Hegen, Martin; Homer, Bruce L; Brodfuehrer, Joanne; Tilley, Mera; Gilbert, Steven A; Danto, Spencer I; Beebe, Jean J; Barnes, Betsy J; Pascual, Virginia; Lin, Lih-Ling; Kilty, Iain; Fleming, Margaret; Rao, Vikram R.
Affiliation
  • Winkler A; Pfizer, Cambridge, Massachusetts.
  • Sun W; Pfizer, Cambridge, Massachusetts.
  • De S; The Feinstein Institute, Manhasset, New York.
  • Jiao A; Pfizer, Cambridge, Massachusetts.
  • Sharif MN; Pfizer, Cambridge, Massachusetts.
  • Symanowicz PT; Pfizer, Cambridge, Massachusetts.
  • Athale S; Baylor Institute for Immunology Research, Dallas, Texas.
  • Shin JH; Pfizer, Cambridge, Massachusetts.
  • Wang J; Pfizer, Cambridge, Massachusetts.
  • Jacobson BA; Pfizer, Cambridge, Massachusetts.
  • Ramsey SJ; Pfizer, Cambridge, Massachusetts.
  • Dower K; Pfizer, Cambridge, Massachusetts.
  • Andreyeva T; Pfizer, Cambridge, Massachusetts.
  • Liu H; Pfizer, Cambridge, Massachusetts.
  • Hegen M; Pfizer, Cambridge, Massachusetts.
  • Homer BL; Pfizer, Cambridge, Massachusetts.
  • Brodfuehrer J; Pfizer, Cambridge, Massachusetts.
  • Tilley M; Pfizer, Cambridge, Massachusetts.
  • Gilbert SA; Pfizer, Cambridge, Massachusetts.
  • Danto SI; Pfizer, Cambridge, Massachusetts.
  • Beebe JJ; Pfizer, Cambridge, Massachusetts.
  • Barnes BJ; The Feinstein Institute, Manhasset, New York.
  • Pascual V; Baylor Institute for Immunology Research, Dallas, Texas.
  • Lin LL; Pfizer, Cambridge, Massachusetts.
  • Kilty I; Pfizer, Cambridge, Massachusetts.
  • Fleming M; Pfizer, Cambridge, Massachusetts.
  • Rao VR; Pfizer, Cambridge, Massachusetts.
Arthritis Rheumatol ; 73(12): 2206-2218, 2021 12.
Article in En | MEDLINE | ID: mdl-34423919

Full text: 1 Database: MEDLINE Main subject: Arthritis, Experimental / Rheumatic Diseases / Interleukin-1 Receptor-Associated Kinases / Synoviocytes / Isoquinolines / Lactams / Macrophages Type of study: Clinical_trials / Risk_factors_studies Limits: Animals / Humans Language: En Journal: Arthritis Rheumatol Year: 2021 Type: Article

Full text: 1 Database: MEDLINE Main subject: Arthritis, Experimental / Rheumatic Diseases / Interleukin-1 Receptor-Associated Kinases / Synoviocytes / Isoquinolines / Lactams / Macrophages Type of study: Clinical_trials / Risk_factors_studies Limits: Animals / Humans Language: En Journal: Arthritis Rheumatol Year: 2021 Type: Article