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Discovery of Selective Tertiary Amide Inhibitors of Cyclin-Dependent Kinase 2 (CDK2).
Zeng, Mingshuo; Grandner, Jessica M; Bryan, Marian C; Verma, Vishal; Larouche-Gauthier, Robin; Leclerc, Jean-Philippe; Zhao, Liang; Haghshenas, Pouyan; Aubert-Nicol, Samuel; Yadav, Arun; Ashley, Melissa; Chen, Jacob Z; Durk, Matthew; Samy, Karen E; Nespi, Marika; Levy, Elizabeth; Merrick, Karl; Moffat, John G; Murray, Jeremy; Oh, Angela; Orr, Christine; Segal, Ehud; Sims, Jessica; Sneeringer, Christopher; Prangley, Madeleine; Vartanian, Steffan; Magnuson, Steven; Parr, Brendan T.
Affiliation
  • Zeng M; Genentech Inc., South San Francisco, California 94080, United States.
  • Grandner JM; Genentech Inc., South San Francisco, California 94080, United States.
  • Bryan MC; Janssen R&D, 1400 McKean Rd, Spring House, Pennsylvania 19002, United States.
  • Verma V; Genentech Inc., South San Francisco, California 94080, United States.
  • Larouche-Gauthier R; Paraza Pharma Inc., Montreal, QC H4S 2E1, Canada.
  • Leclerc JP; Paraza Pharma Inc., Montreal, QC H4S 2E1, Canada.
  • Zhao L; Paraza Pharma Inc., Montreal, QC H4S 2E1, Canada.
  • Haghshenas P; Paraza Pharma Inc., Montreal, QC H4S 2E1, Canada.
  • Aubert-Nicol S; Paraza Pharma Inc., Montreal, QC H4S 2E1, Canada.
  • Yadav A; Paraza Pharma Inc., Montreal, QC H4S 2E1, Canada.
  • Ashley M; Genentech Inc., South San Francisco, California 94080, United States.
  • Chen JZ; Genentech Inc., South San Francisco, California 94080, United States.
  • Durk M; Genentech Inc., South San Francisco, California 94080, United States.
  • Samy KE; Genentech Inc., South San Francisco, California 94080, United States.
  • Nespi M; Genentech Inc., South San Francisco, California 94080, United States.
  • Levy E; Genentech Inc., South San Francisco, California 94080, United States.
  • Merrick K; Genentech Inc., South San Francisco, California 94080, United States.
  • Moffat JG; Genentech Inc., South San Francisco, California 94080, United States.
  • Murray J; Genentech Inc., South San Francisco, California 94080, United States.
  • Oh A; Genentech Inc., South San Francisco, California 94080, United States.
  • Orr C; Genentech Inc., South San Francisco, California 94080, United States.
  • Segal E; Genentech Inc., South San Francisco, California 94080, United States.
  • Sims J; Genentech Inc., South San Francisco, California 94080, United States.
  • Sneeringer C; Genentech Inc., South San Francisco, California 94080, United States.
  • Prangley M; Genentech Inc., South San Francisco, California 94080, United States.
  • Vartanian S; Genentech Inc., South San Francisco, California 94080, United States.
  • Magnuson S; Genentech Inc., South San Francisco, California 94080, United States.
  • Parr BT; Genentech Inc., South San Francisco, California 94080, United States.
ACS Med Chem Lett ; 14(9): 1179-1187, 2023 Sep 14.
Article in En | MEDLINE | ID: mdl-37736184

Full text: 1 Database: MEDLINE Language: En Journal: ACS Med Chem Lett Year: 2023 Type: Article Affiliation country: United States

Full text: 1 Database: MEDLINE Language: En Journal: ACS Med Chem Lett Year: 2023 Type: Article Affiliation country: United States