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Optimization of 2-Anilino 4-Amino Substituted Quinazolines into Potent Antimalarial Agents with Oral in Vivo Activity.
Gilson, Paul R; Tan, Cyrus; Jarman, Kate E; Lowes, Kym N; Curtis, Joan M; Nguyen, William; Di Rago, Adrian E; Bullen, Hayley E; Prinz, Boris; Duffy, Sandra; Baell, Jonathan B; Hutton, Craig A; Jousset Subroux, Helene; Crabb, Brendan S; Avery, Vicky M; Cowman, Alan F; Sleebs, Brad E.
Afiliación
  • Gilson PR; Macfarlane Burnet Institute for Medical Research and Public Health , Melbourne, 3004, Australia.
  • Tan C; Monash University , Clayton, Victoria 3800, Australia.
  • Jarman KE; The Walter and Eliza Hall Institute of Medical Research , Parkville 3052, Australia.
  • Lowes KN; Department of Medical Biology, The University of Melbourne , Parkville 3010, Australia.
  • Curtis JM; The Walter and Eliza Hall Institute of Medical Research , Parkville 3052, Australia.
  • Nguyen W; Department of Medical Biology, The University of Melbourne , Parkville 3010, Australia.
  • Di Rago AE; The Walter and Eliza Hall Institute of Medical Research , Parkville 3052, Australia.
  • Bullen HE; Department of Medical Biology, The University of Melbourne , Parkville 3010, Australia.
  • Prinz B; The Walter and Eliza Hall Institute of Medical Research , Parkville 3052, Australia.
  • Duffy S; The Walter and Eliza Hall Institute of Medical Research , Parkville 3052, Australia.
  • Baell JB; Department of Medical Biology, The University of Melbourne , Parkville 3010, Australia.
  • Hutton CA; The Walter and Eliza Hall Institute of Medical Research , Parkville 3052, Australia.
  • Jousset Subroux H; Macfarlane Burnet Institute for Medical Research and Public Health , Melbourne, 3004, Australia.
  • Crabb BS; Macfarlane Burnet Institute for Medical Research and Public Health , Melbourne, 3004, Australia.
  • Avery VM; Discovery Biology, Eskitis Institute for Drug Discovery, Griffith University , Nathan, Queensland 4111, Australia.
  • Cowman AF; Monash Institute of Pharmaceutical Sciences, Monash University , Parkville, Victoria 3052, Australia.
  • Sleebs BE; School of Chemistry and Bio21 Molecular Science and Biotechnology Institute, University of Melbourne , Parkville, Victoria 3010, Australia.
J Med Chem ; 60(3): 1171-1188, 2017 02 09.
Article en En | MEDLINE | ID: mdl-28080063

Texto completo: 1 Bases de datos: MEDLINE Asunto principal: Quinazolinas / Antimaláricos Límite: Animals Idioma: En Revista: J Med Chem Asunto de la revista: QUIMICA Año: 2017 Tipo del documento: Article País de afiliación: Australia

Texto completo: 1 Bases de datos: MEDLINE Asunto principal: Quinazolinas / Antimaláricos Límite: Animals Idioma: En Revista: J Med Chem Asunto de la revista: QUIMICA Año: 2017 Tipo del documento: Article País de afiliación: Australia