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Exploration of ligand binding modes towards the identification of compounds targeting HuR: a combined STD-NMR and Molecular Modelling approach.
Vasile, Francesca; Della Volpe, Serena; Ambrosio, Francesca Alessandra; Costa, Giosuè; Unver, M Yagiz; Zucal, Chiara; Rossi, Daniela; Martino, Emanuela; Provenzani, Alessandro; Hirsch, Anna K H; Alcaro, Stefano; Potenza, Donatella; Collina, Simona.
Afiliación
  • Vasile F; Department of Chemistry, University of Milan, Via Golgi 19, 20133, Milano, Italy.
  • Della Volpe S; Department of Chemistry, University of Milan, Via Golgi 19, 20133, Milano, Italy.
  • Ambrosio FA; Department of Drug Sciences, Medicinal Chemistry and Technology Section, University of Pavia, Via Taramelli 12, 27100, Pavia, Italy.
  • Costa G; Department of Health Sciences, University "Magna Græcia" of Catanzaro, Viale Europa, 88100, Catanzaro, Italy.
  • Unver MY; Department of Health Sciences, University "Magna Græcia" of Catanzaro, Viale Europa, 88100, Catanzaro, Italy.
  • Zucal C; Helmholtz Institute for Pharmaceutical Research Saarland (HIPS) - Helmholtz Centre for Infection Research (HZI), Department of Drug Design and Optimization, Campus building E8.1, 66123, Saarbrücken, Germany.
  • Rossi D; Centre for Integrative Biology, CIBIO, University of Trento, Via Sommarive 9, 38123, Povo, TN, Italy.
  • Martino E; Department of Drug Sciences, Medicinal Chemistry and Technology Section, University of Pavia, Via Taramelli 12, 27100, Pavia, Italy.
  • Provenzani A; Department of Earth and Environmental Sciences, University of Pavia, via S. Epifanio 14, 27100, Pavia, Italy.
  • Hirsch AKH; Centre for Integrative Biology, CIBIO, University of Trento, Via Sommarive 9, 38123, Povo, TN, Italy.
  • Alcaro S; Helmholtz Institute for Pharmaceutical Research Saarland (HIPS) - Helmholtz Centre for Infection Research (HZI), Department of Drug Design and Optimization, Campus building E8.1, 66123, Saarbrücken, Germany.
  • Potenza D; Department of Pharmacy, Medicinal Chemistry, Saarland University, Campus building E8.1, 66123, Saarbrücken, Germany.
  • Collina S; Department of Health Sciences, University "Magna Græcia" of Catanzaro, Viale Europa, 88100, Catanzaro, Italy.
Sci Rep ; 8(1): 13780, 2018 09 13.
Article en En | MEDLINE | ID: mdl-30214075

Texto completo: 1 Bases de datos: MEDLINE Asunto principal: Flavonoides / Procesamiento Postranscripcional del ARN / Regulación de la Expresión Génica / Cumarinas / Proteína 1 Similar a ELAV Tipo de estudio: Diagnostic_studies Límite: Humans Idioma: En Revista: Sci Rep Año: 2018 Tipo del documento: Article País de afiliación: Italia

Texto completo: 1 Bases de datos: MEDLINE Asunto principal: Flavonoides / Procesamiento Postranscripcional del ARN / Regulación de la Expresión Génica / Cumarinas / Proteína 1 Similar a ELAV Tipo de estudio: Diagnostic_studies Límite: Humans Idioma: En Revista: Sci Rep Año: 2018 Tipo del documento: Article País de afiliación: Italia