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Studies on the inhibition of AmpC and other ß-lactamases by cyclic boronates.
Cahill, Samuel T; Tyrrell, Jonathan M; Navratilova, Iva Hopkins; Calvopiña, Karina; Robinson, Sean W; Lohans, Christopher T; McDonough, Michael A; Cain, Ricky; Fishwick, Colin W G; Avison, Matthew B; Walsh, Timothy R; Schofield, Christopher J; Brem, Jürgen.
Afiliación
  • Cahill ST; Department of Chemistry, University of Oxford, Chemistry Research Laboratory, 12 Mansfield Road, Oxford OX1 3TA, United Kingdom.
  • Tyrrell JM; Department of Medical Microbiology & Infectious Disease, Institute of Infection & Immunity, UHW Main Building, Heath Park, Cardiff CF14 4XN, United Kingdom.
  • Navratilova IH; University of Dundee, Dow Street, Dundee DD1 5EH, United Kingdom; Research Complex at Harwell, Rutherford Appleton Lab, Harwell, Oxford OX11 0FA, United Kingdom.
  • Calvopiña K; School of Cellular and Molecular Medicine, University of Bristol, Biomedical Sciences Building, Bristol BS8 1TD, United Kingdom.
  • Robinson SW; Kinetic Discovery Ltd, Rutherford Appleton Laboratory, Oxford, Didcot OX11 0FA, United Kingdom.
  • Lohans CT; Department of Chemistry, University of Oxford, Chemistry Research Laboratory, 12 Mansfield Road, Oxford OX1 3TA, United Kingdom.
  • McDonough MA; Department of Chemistry, University of Oxford, Chemistry Research Laboratory, 12 Mansfield Road, Oxford OX1 3TA, United Kingdom.
  • Cain R; School of Chemistry, University of Leeds, Leeds LS2 9JT, United Kingdom.
  • Fishwick CWG; School of Chemistry, University of Leeds, Leeds LS2 9JT, United Kingdom.
  • Avison MB; School of Cellular and Molecular Medicine, University of Bristol, Biomedical Sciences Building, Bristol BS8 1TD, United Kingdom.
  • Walsh TR; Department of Medical Microbiology & Infectious Disease, Institute of Infection & Immunity, UHW Main Building, Heath Park, Cardiff CF14 4XN, United Kingdom.
  • Schofield CJ; Department of Chemistry, University of Oxford, Chemistry Research Laboratory, 12 Mansfield Road, Oxford OX1 3TA, United Kingdom. Electronic address: christopher.schofield@chem.ox.ac.uk.
  • Brem J; Department of Chemistry, University of Oxford, Chemistry Research Laboratory, 12 Mansfield Road, Oxford OX1 3TA, United Kingdom. Electronic address: jurgen.brem@chem.ox.ac.uk.
Biochim Biophys Acta Gen Subj ; 1863(4): 742-748, 2019 04.
Article en En | MEDLINE | ID: mdl-30738906

Texto completo: 1 Bases de datos: MEDLINE Asunto principal: Beta-Lactamasas / Ácidos Borónicos / Inhibidores de beta-Lactamasas / Antibacterianos Idioma: En Revista: Biochim Biophys Acta Gen Subj Año: 2019 Tipo del documento: Article País de afiliación: Reino Unido

Texto completo: 1 Bases de datos: MEDLINE Asunto principal: Beta-Lactamasas / Ácidos Borónicos / Inhibidores de beta-Lactamasas / Antibacterianos Idioma: En Revista: Biochim Biophys Acta Gen Subj Año: 2019 Tipo del documento: Article País de afiliación: Reino Unido