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Search for multifunctional agents against Alzheimer's disease among non-imidazole histamine H3 receptor ligands. In vitro and in vivo pharmacological evaluation and computational studies of piperazine derivatives.
Jonczyk, Jakub; Lodarski, Krzysztof; Staszewski, Marek; Godyn, Justyna; Zareba, Paula; Soukup, Ondrej; Janockova, Jana; Korabecny, Jan; Salat, Kinga; Malikowska-Racia, Natalia; Hebda, Michalina; Szalaj, Natalia; Filipek, Barbara; Walczynski, Krzysztof; Malawska, Barbara; Bajda, Marek.
Afiliación
  • Jonczyk J; Department of Physicochemical Drug Analysis, Faculty of Pharmacy, Jagiellonian University Medical College, Medyczna 9, 30-688 Kraków, Poland.
  • Lodarski K; Department of Physicochemical Drug Analysis, Faculty of Pharmacy, Jagiellonian University Medical College, Medyczna 9, 30-688 Kraków, Poland.
  • Staszewski M; Department of Synthesis and Technology of Drugs, Medical University of Lódz, Muszynskiego 1, 90-145 Lódz, Poland.
  • Godyn J; Department of Physicochemical Drug Analysis, Faculty of Pharmacy, Jagiellonian University Medical College, Medyczna 9, 30-688 Kraków, Poland.
  • Zareba P; Department of Physicochemical Drug Analysis, Faculty of Pharmacy, Jagiellonian University Medical College, Medyczna 9, 30-688 Kraków, Poland.
  • Soukup O; Biomedical Research Center, University Hospital Hradec Kralove, Sokolska 581, 500 05 Hradec Kralove, Czech Republic; National Institute of Mental Health, Topolova 748, 250 67 Klecany, Czech Republic.
  • Janockova J; Biomedical Research Center, University Hospital Hradec Kralove, Sokolska 581, 500 05 Hradec Kralove, Czech Republic.
  • Korabecny J; Biomedical Research Center, University Hospital Hradec Kralove, Sokolska 581, 500 05 Hradec Kralove, Czech Republic; National Institute of Mental Health, Topolova 748, 250 67 Klecany, Czech Republic.
  • Salat K; Department of Pharmacodynamics, Jagiellonian University Medical College, Medyczna 9, 30-688 Kraków, Poland.
  • Malikowska-Racia N; Department of Pharmacodynamics, Jagiellonian University Medical College, Medyczna 9, 30-688 Kraków, Poland.
  • Hebda M; Department of Physicochemical Drug Analysis, Faculty of Pharmacy, Jagiellonian University Medical College, Medyczna 9, 30-688 Kraków, Poland.
  • Szalaj N; Department of Physicochemical Drug Analysis, Faculty of Pharmacy, Jagiellonian University Medical College, Medyczna 9, 30-688 Kraków, Poland.
  • Filipek B; Department of Pharmacodynamics, Jagiellonian University Medical College, Medyczna 9, 30-688 Kraków, Poland.
  • Walczynski K; Department of Synthesis and Technology of Drugs, Medical University of Lódz, Muszynskiego 1, 90-145 Lódz, Poland.
  • Malawska B; Department of Physicochemical Drug Analysis, Faculty of Pharmacy, Jagiellonian University Medical College, Medyczna 9, 30-688 Kraków, Poland.
  • Bajda M; Department of Physicochemical Drug Analysis, Faculty of Pharmacy, Jagiellonian University Medical College, Medyczna 9, 30-688 Kraków, Poland. Electronic address: marek.bajda@uj.edu.pl.
Bioorg Chem ; 90: 103084, 2019 09.
Article en En | MEDLINE | ID: mdl-31271942

Texto completo: 1 Bases de datos: MEDLINE Asunto principal: Piperazinas / Inhibidores de la Colinesterasa / Receptores Histamínicos H3 / Modelos Animales de Enfermedad / Enfermedad de Alzheimer / Amnesia Tipo de estudio: Evaluation_studies Límite: Animals Idioma: En Revista: Bioorg Chem Año: 2019 Tipo del documento: Article País de afiliación: Polonia

Texto completo: 1 Bases de datos: MEDLINE Asunto principal: Piperazinas / Inhibidores de la Colinesterasa / Receptores Histamínicos H3 / Modelos Animales de Enfermedad / Enfermedad de Alzheimer / Amnesia Tipo de estudio: Evaluation_studies Límite: Animals Idioma: En Revista: Bioorg Chem Año: 2019 Tipo del documento: Article País de afiliación: Polonia