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Allosteric inhibitors of Mycobacterium tuberculosis tryptophan synthase.
Michalska, Karolina; Chang, Changsoo; Maltseva, Natalia I; Jedrzejczak, Robert; Robertson, Gregory T; Gusovsky, Fabian; McCarren, Patrick; Schreiber, Stuart L; Nag, Partha P; Joachimiak, Andrzej.
Afiliación
  • Michalska K; Center for Structural Genomics of Infectious Diseases, Consortium for Advanced Science and Engineering, University of Chicago, Chicago, Illinois.
  • Chang C; Structural Biology Center, X-ray Science Division, Argonne National Laboratory, Argonne, Illinois.
  • Maltseva NI; Center for Structural Genomics of Infectious Diseases, Consortium for Advanced Science and Engineering, University of Chicago, Chicago, Illinois.
  • Jedrzejczak R; Structural Biology Center, X-ray Science Division, Argonne National Laboratory, Argonne, Illinois.
  • Robertson GT; Center for Structural Genomics of Infectious Diseases, Consortium for Advanced Science and Engineering, University of Chicago, Chicago, Illinois.
  • Gusovsky F; Structural Biology Center, X-ray Science Division, Argonne National Laboratory, Argonne, Illinois.
  • McCarren P; Center for Structural Genomics of Infectious Diseases, Consortium for Advanced Science and Engineering, University of Chicago, Chicago, Illinois.
  • Schreiber SL; Structural Biology Center, X-ray Science Division, Argonne National Laboratory, Argonne, Illinois.
  • Nag PP; Colorado State University, Mycobacteria Research Laboratories, Department of Microbiology, Immunology and Pathology, Fort Collins, Colorado.
  • Joachimiak A; Eisai Co, Ltd., World Health Initiative, Andover, Massachusetts.
Protein Sci ; 29(3): 779-788, 2020 03.
Article en En | MEDLINE | ID: mdl-31930594

Texto completo: 1 Bases de datos: MEDLINE Asunto principal: Sulfonamidas / Tiofenos / Triptófano Sintasa / Inhibidores Enzimáticos / Sitio Alostérico / Indoles / Mycobacterium tuberculosis Tipo de estudio: Prognostic_studies Límite: Humans Idioma: En Revista: Protein Sci Asunto de la revista: BIOQUIMICA Año: 2020 Tipo del documento: Article

Texto completo: 1 Bases de datos: MEDLINE Asunto principal: Sulfonamidas / Tiofenos / Triptófano Sintasa / Inhibidores Enzimáticos / Sitio Alostérico / Indoles / Mycobacterium tuberculosis Tipo de estudio: Prognostic_studies Límite: Humans Idioma: En Revista: Protein Sci Asunto de la revista: BIOQUIMICA Año: 2020 Tipo del documento: Article