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Structure-Activity Relationships of Noncovalent Immunoproteasome ß5i-Selective Dipeptides.
Zhan, Wenhu; Singh, Pradeep K; Ban, Yi; Qing, Xiaoping; Ah Kioon, Marie Dominique; Fan, Hao; Zhao, Quanju; Wang, Rong; Sukenick, George; Salmon, Jane; Warren, J David; Ma, Xiaojing; Barrat, Franck J; Nathan, Carl F; Lin, Gang.
Afiliación
  • Zhan W; Department of Microbiology & Immunology, Weill Cornell Medicine, 1300 York Ave, New York, New York 10065, United States.
  • Singh PK; Department of Biochemistry, Milstein Chemistry Core Facility, Weill Cornell Medicine, 1300 York Ave, New York, New York 10065, United States.
  • Ban Y; Department of Microbiology & Immunology, Weill Cornell Medicine, 1300 York Ave, New York, New York 10065, United States.
  • Qing X; Autoimmunity and Inflammation Program, HSS Research Institute, Hospital for Special Surgery, New York, New York 10065, United States.
  • Ah Kioon MD; Autoimmunity and Inflammation Program, HSS Research Institute, Hospital for Special Surgery, New York, New York 10065, United States.
  • Fan H; Department of Microbiology & Immunology, Weill Cornell Medicine, 1300 York Ave, New York, New York 10065, United States.
  • Zhao Q; Department of Microbiology & Immunology, Weill Cornell Medicine, 1300 York Ave, New York, New York 10065, United States.
  • Wang R; NMR Analytical Core Facility, Memorial Sloan Kettering Cancer Center, 417 East 68th Street, Room 1735, New York, New York 10065-6007, United States.
  • Sukenick G; NMR Analytical Core Facility, Memorial Sloan Kettering Cancer Center, 417 East 68th Street, Room 1735, New York, New York 10065-6007, United States.
  • Salmon J; Autoimmunity and Inflammation Program, HSS Research Institute, Hospital for Special Surgery, New York, New York 10065, United States.
  • Warren JD; Department of Biochemistry, Milstein Chemistry Core Facility, Weill Cornell Medicine, 1300 York Ave, New York, New York 10065, United States.
  • Ma X; Department of Microbiology & Immunology, Weill Cornell Medicine, 1300 York Ave, New York, New York 10065, United States.
  • Barrat FJ; Department of Microbiology & Immunology, Weill Cornell Medicine, 1300 York Ave, New York, New York 10065, United States.
  • Nathan CF; Autoimmunity and Inflammation Program, HSS Research Institute, Hospital for Special Surgery, New York, New York 10065, United States.
  • Lin G; Department of Microbiology & Immunology, Weill Cornell Medicine, 1300 York Ave, New York, New York 10065, United States.
J Med Chem ; 63(21): 13103-13123, 2020 11 12.
Article en En | MEDLINE | ID: mdl-33095579

Texto completo: 1 Bases de datos: MEDLINE Asunto principal: Complejo de la Endopetidasa Proteasomal / Dipéptidos / Inhibidores de Proteasoma Límite: Humans Idioma: En Revista: J Med Chem Asunto de la revista: QUIMICA Año: 2020 Tipo del documento: Article País de afiliación: Estados Unidos

Texto completo: 1 Bases de datos: MEDLINE Asunto principal: Complejo de la Endopetidasa Proteasomal / Dipéptidos / Inhibidores de Proteasoma Límite: Humans Idioma: En Revista: J Med Chem Asunto de la revista: QUIMICA Año: 2020 Tipo del documento: Article País de afiliación: Estados Unidos