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Synthesis and Biological Activity of a Cytostatic Inhibitor of MLLr Leukemia Targeting the DOT1L Protein.
Bon, Corentin; Si, Yang; Pernak, Melanie; Barbachowska, Magdalena; Levi-Acobas, Eva; Cadet Daniel, Veronique; Jallet, Corinne; Ruzic, Dusan; Djokovic, Nemanja; Djikic, Teodora; Nikolic, Katarina; Halby, Ludovic; Arimondo, Paola B.
Afiliación
  • Bon C; Epigenetic Chemical Biology, Department of Structural Biology and Chemistry, Institut Pasteur, UMR3523 CNRS, 75015 Paris, France.
  • Si Y; Ecole Doctorale MTCI, Université de Paris, Sorbonne Paris Cité, 75006 Paris, France.
  • Pernak M; Epigenetic Chemical Biology, Department of Structural Biology and Chemistry, Institut Pasteur, UMR3523 CNRS, 75015 Paris, France.
  • Barbachowska M; Epigenetic Chemical Biology, Department of Structural Biology and Chemistry, Institut Pasteur, UMR3523 CNRS, 75015 Paris, France.
  • Levi-Acobas E; Epigenetic Chemical Biology, Department of Structural Biology and Chemistry, Institut Pasteur, UMR3523 CNRS, 75015 Paris, France.
  • Cadet Daniel V; Ecole Doctorale MTCI, Université de Paris, Sorbonne Paris Cité, 75006 Paris, France.
  • Jallet C; Epigenetic Chemical Biology, Department of Structural Biology and Chemistry, Institut Pasteur, UMR3523 CNRS, 75015 Paris, France.
  • Ruzic D; Epigenetic Chemical Biology, Department of Structural Biology and Chemistry, Institut Pasteur, UMR3523 CNRS, 75015 Paris, France.
  • Djokovic N; Epigenetic Chemical Biology, Department of Structural Biology and Chemistry, Institut Pasteur, UMR3523 CNRS, 75015 Paris, France.
  • Djikic T; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, University of Belgrade, Vojvode Stepe 450, 11000 Belgrade, Serbia.
  • Nikolic K; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, University of Belgrade, Vojvode Stepe 450, 11000 Belgrade, Serbia.
  • Halby L; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, University of Belgrade, Vojvode Stepe 450, 11000 Belgrade, Serbia.
  • Arimondo PB; Department of Pharmaceutical Chemistry, Faculty of Pharmacy, University of Belgrade, Vojvode Stepe 450, 11000 Belgrade, Serbia.
Molecules ; 26(17)2021 Aug 31.
Article en En | MEDLINE | ID: mdl-34500733

Texto completo: 1 Bases de datos: MEDLINE Asunto principal: Histonas / N-Metiltransferasa de Histona-Lisina / Citostáticos Límite: Humans Idioma: En Revista: Molecules Asunto de la revista: BIOLOGIA Año: 2021 Tipo del documento: Article País de afiliación: Francia

Texto completo: 1 Bases de datos: MEDLINE Asunto principal: Histonas / N-Metiltransferasa de Histona-Lisina / Citostáticos Límite: Humans Idioma: En Revista: Molecules Asunto de la revista: BIOLOGIA Año: 2021 Tipo del documento: Article País de afiliación: Francia