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Insights Into Drug Repurposing, as Well as Specificity and Compound Properties of Piperidine-Based SARS-CoV-2 PLpro Inhibitors.
Calleja, Dale J; Kuchel, Nathan; Lu, Bernadine G C; Birkinshaw, Richard W; Klemm, Theresa; Doerflinger, Marcel; Cooney, James P; Mackiewicz, Liana; Au, Amanda E; Yap, Yu Q; Blackmore, Timothy R; Katneni, Kasiram; Crighton, Elly; Newman, Janet; Jarman, Kate E; Call, Melissa J; Lechtenberg, Bernhard C; Czabotar, Peter E; Pellegrini, Marc; Charman, Susan A; Lowes, Kym N; Mitchell, Jeffrey P; Nachbur, Ueli; Lessene, Guillaume; Komander, David.
Afiliación
  • Calleja DJ; Department of Medical Biology, Walter and Eliza Hall Institute, University of Melbourne, Melbourne, VIC, Australia.
  • Kuchel N; Department of Medical Biology, Walter and Eliza Hall Institute, University of Melbourne, Melbourne, VIC, Australia.
  • Lu BGC; Department of Medical Biology, Walter and Eliza Hall Institute, University of Melbourne, Melbourne, VIC, Australia.
  • Birkinshaw RW; Department of Medical Biology, Walter and Eliza Hall Institute, University of Melbourne, Melbourne, VIC, Australia.
  • Klemm T; Department of Medical Biology, Walter and Eliza Hall Institute, University of Melbourne, Melbourne, VIC, Australia.
  • Doerflinger M; Department of Medical Biology, Walter and Eliza Hall Institute, University of Melbourne, Melbourne, VIC, Australia.
  • Cooney JP; Department of Medical Biology, Walter and Eliza Hall Institute, University of Melbourne, Melbourne, VIC, Australia.
  • Mackiewicz L; Department of Medical Biology, Walter and Eliza Hall Institute, University of Melbourne, Melbourne, VIC, Australia.
  • Au AE; Department of Medical Biology, Walter and Eliza Hall Institute, University of Melbourne, Melbourne, VIC, Australia.
  • Yap YQ; Department of Medical Biology, Walter and Eliza Hall Institute, University of Melbourne, Melbourne, VIC, Australia.
  • Blackmore TR; Department of Medical Biology, Walter and Eliza Hall Institute, University of Melbourne, Melbourne, VIC, Australia.
  • Katneni K; Centre for Drug Candidate Optimisation, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, VIC, Australia.
  • Crighton E; Centre for Drug Candidate Optimisation, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, VIC, Australia.
  • Newman J; Commonwealth Scientific and Industrial Research Organisation (CSIRO), Biomedical Program, Parkville, VIC, Australia.
  • Jarman KE; Department of Medical Biology, Walter and Eliza Hall Institute, University of Melbourne, Melbourne, VIC, Australia.
  • Call MJ; Department of Medical Biology, Walter and Eliza Hall Institute, University of Melbourne, Melbourne, VIC, Australia.
  • Lechtenberg BC; Department of Medical Biology, Walter and Eliza Hall Institute, University of Melbourne, Melbourne, VIC, Australia.
  • Czabotar PE; Department of Medical Biology, Walter and Eliza Hall Institute, University of Melbourne, Melbourne, VIC, Australia.
  • Pellegrini M; Department of Medical Biology, Walter and Eliza Hall Institute, University of Melbourne, Melbourne, VIC, Australia.
  • Charman SA; Centre for Drug Candidate Optimisation, Monash Institute of Pharmaceutical Sciences, Monash University, Parkville, VIC, Australia.
  • Lowes KN; Department of Medical Biology, Walter and Eliza Hall Institute, University of Melbourne, Melbourne, VIC, Australia.
  • Mitchell JP; Department of Medical Biology, Walter and Eliza Hall Institute, University of Melbourne, Melbourne, VIC, Australia.
  • Nachbur U; Department of Medical Biology, Walter and Eliza Hall Institute, University of Melbourne, Melbourne, VIC, Australia.
  • Lessene G; Department of Medical Biology, Walter and Eliza Hall Institute, University of Melbourne, Melbourne, VIC, Australia.
  • Komander D; Department of Pharmacology and Therapeutics, The University of Melbourne, Melbourne, VIC, Australia.
Front Chem ; 10: 861209, 2022.
Article en En | MEDLINE | ID: mdl-35494659

Texto completo: 1 Bases de datos: MEDLINE Tipo de estudio: Prognostic_studies Idioma: En Revista: Front Chem Año: 2022 Tipo del documento: Article País de afiliación: Australia

Texto completo: 1 Bases de datos: MEDLINE Tipo de estudio: Prognostic_studies Idioma: En Revista: Front Chem Año: 2022 Tipo del documento: Article País de afiliación: Australia