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Design and synthesis of harmiquins, harmine and chloroquine hybrids as potent antiplasmodial agents.
Poje, Goran; Pessanha de Carvalho, Lais; Held, Jana; Moita, Diana; Prudêncio, Miguel; Perkovic, Ivana; Tandaric, Tana; Vianello, Robert; Rajic, Zrinka.
Afiliación
  • Poje G; University of Zagreb Faculty of Pharmacy and Biochemistry, A. Kovacica 1, 10000, Zagreb, Croatia.
  • Pessanha de Carvalho L; University of Tübingen, Institute of Tropical Medicine, Wilhelmstraße 27, 72074, Tübingen, Germany.
  • Held J; University of Tübingen, Institute of Tropical Medicine, Wilhelmstraße 27, 72074, Tübingen, Germany; German Center for Infection Research (DZIF), Partner Site Tübingen, 72074, Tübingen, Germany.
  • Moita D; Instituto de Medicina Molecular João Lobo Antunes, Faculdade de Medicina, Universidade de Lisboa, Av. Prof. Egas Moniz, 1649-028, Lisboa, Portugal.
  • Prudêncio M; Instituto de Medicina Molecular João Lobo Antunes, Faculdade de Medicina, Universidade de Lisboa, Av. Prof. Egas Moniz, 1649-028, Lisboa, Portugal.
  • Perkovic I; University of Zagreb Faculty of Pharmacy and Biochemistry, A. Kovacica 1, 10000, Zagreb, Croatia.
  • Tandaric T; Rudjer Boskovic Institute, Division of Organic Chemistry and Biochemistry, Bijenicka cesta 54, 10 000, Zagreb, Croatia.
  • Vianello R; Rudjer Boskovic Institute, Division of Organic Chemistry and Biochemistry, Bijenicka cesta 54, 10 000, Zagreb, Croatia.
  • Rajic Z; University of Zagreb Faculty of Pharmacy and Biochemistry, A. Kovacica 1, 10000, Zagreb, Croatia. Electronic address: zrajic@pharma.hr.
Eur J Med Chem ; 238: 114408, 2022 Aug 05.
Article en En | MEDLINE | ID: mdl-35551033

Texto completo: 1 Bases de datos: MEDLINE Asunto principal: Malaria Falciparum / Antimaláricos Límite: Humans Idioma: En Revista: Eur J Med Chem Año: 2022 Tipo del documento: Article País de afiliación: Croacia

Texto completo: 1 Bases de datos: MEDLINE Asunto principal: Malaria Falciparum / Antimaláricos Límite: Humans Idioma: En Revista: Eur J Med Chem Año: 2022 Tipo del documento: Article País de afiliación: Croacia