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ΔF508-CFTR correctors: synthesis and evaluation of thiazole-tethered imidazolones, oxazoles, oxadiazoles, and thiadiazoles.
Ye, Long; Hu, Bao; El-Badri, Faris; Hudson, Brandi M; Phuan, Puay-Wah; Verkman, A S; Tantillo, Dean J; Kurth, Mark J.
Afiliação
  • Ye L; Department of Chemistry, College of Chemical Engineering and Technology, Wuhan University of Science and Technology, Wuhan, Hubei 430081, PR China. Electronic address: yelong@wust.edu.cn.
  • Hu B; Department of Chemistry, College of Chemical Engineering and Technology, Wuhan University of Science and Technology, Wuhan, Hubei 430081, PR China.
  • El-Badri F; Department of Chemistry, University of California, One Shields Ave, Davis, CA 95616, United States.
  • Hudson BM; Department of Chemistry, University of California, One Shields Ave, Davis, CA 95616, United States.
  • Phuan PW; Department of Medicine, University of California, San Francisco, CA 94143-0521, United States; Department Physiology, University of California, San Francisco, CA 94143-0521, United States.
  • Verkman AS; Department of Medicine, University of California, San Francisco, CA 94143-0521, United States; Department Physiology, University of California, San Francisco, CA 94143-0521, United States.
  • Tantillo DJ; Department of Chemistry, University of California, One Shields Ave, Davis, CA 95616, United States.
  • Kurth MJ; Department of Chemistry, University of California, One Shields Ave, Davis, CA 95616, United States. Electronic address: mjkurth@ucdavis.edu.
Bioorg Med Chem Lett ; 24(24): 5840-5844, 2014 Dec 15.
Article em En | MEDLINE | ID: mdl-25452003

Texto completo: 1 Bases de dados: MEDLINE Assunto principal: Oxidiazóis / Oxazóis / Tiadiazóis / Regulador de Condutância Transmembrana em Fibrose Cística / Imidazóis Limite: Humans Idioma: En Revista: Bioorg Med Chem Lett Assunto da revista: BIOQUIMICA / QUIMICA Ano de publicação: 2014 Tipo de documento: Article

Texto completo: 1 Bases de dados: MEDLINE Assunto principal: Oxidiazóis / Oxazóis / Tiadiazóis / Regulador de Condutância Transmembrana em Fibrose Cística / Imidazóis Limite: Humans Idioma: En Revista: Bioorg Med Chem Lett Assunto da revista: BIOQUIMICA / QUIMICA Ano de publicação: 2014 Tipo de documento: Article