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Discovery of 6-phenylimidazo[2,1-b]thiazole derivatives as a new type of FLT3 inhibitors.
Lin, Xing-Dong; Yang, Hui-Wen; Ma, Shuang; Li, Wei-Wei; Zhang, Chun-Hui; Wang, Wen-Jing; Xiang, Rong; Li, Lin-Li; Yang, Sheng-Yong.
Afiliação
  • Lin XD; State Key Laboratory of Biotherapy and Cancer Center, West China Hospital, Sichuan University, and Collaborative Innovation Center for Biotherapy, Sichuan 610041, China.
  • Yang HW; State Key Laboratory of Biotherapy and Cancer Center, West China Hospital, Sichuan University, and Collaborative Innovation Center for Biotherapy, Sichuan 610041, China.
  • Ma S; State Key Laboratory of Biotherapy and Cancer Center, West China Hospital, Sichuan University, and Collaborative Innovation Center for Biotherapy, Sichuan 610041, China.
  • Li WW; State Key Laboratory of Biotherapy and Cancer Center, West China Hospital, Sichuan University, and Collaborative Innovation Center for Biotherapy, Sichuan 610041, China.
  • Zhang CH; State Key Laboratory of Biotherapy and Cancer Center, West China Hospital, Sichuan University, and Collaborative Innovation Center for Biotherapy, Sichuan 610041, China.
  • Wang WJ; State Key Laboratory of Biotherapy and Cancer Center, West China Hospital, Sichuan University, and Collaborative Innovation Center for Biotherapy, Sichuan 610041, China.
  • Xiang R; Department of Clinical Medicine, School of Medicine, Nankai University, Tianjin, China.
  • Li LL; West China School of Pharmacy, Sichuan University, Sichuan 610041, China. Electronic address: ysylilinli@sina.com.cn.
  • Yang SY; State Key Laboratory of Biotherapy and Cancer Center, West China Hospital, Sichuan University, and Collaborative Innovation Center for Biotherapy, Sichuan 610041, China. Electronic address: yangsy@scu.edu.cn.
Bioorg Med Chem Lett ; 25(20): 4534-8, 2015 Oct 15.
Article em En | MEDLINE | ID: mdl-26342867

Texto completo: 1 Bases de dados: MEDLINE Assunto principal: Compostos de Fenilureia / Tiazóis / Inibidores de Proteínas Quinases / Tirosina Quinase 3 Semelhante a fms / Descoberta de Drogas Limite: Humans Idioma: En Revista: Bioorg Med Chem Lett Assunto da revista: BIOQUIMICA / QUIMICA Ano de publicação: 2015 Tipo de documento: Article País de afiliação: China

Texto completo: 1 Bases de dados: MEDLINE Assunto principal: Compostos de Fenilureia / Tiazóis / Inibidores de Proteínas Quinases / Tirosina Quinase 3 Semelhante a fms / Descoberta de Drogas Limite: Humans Idioma: En Revista: Bioorg Med Chem Lett Assunto da revista: BIOQUIMICA / QUIMICA Ano de publicação: 2015 Tipo de documento: Article País de afiliação: China