Your browser doesn't support javascript.
loading
Discovery of the First α-Amino-3-hydroxy-5-methyl-4-isoxazolepropionic Acid (AMPA) Receptor Antagonist Dependent upon Transmembrane AMPA Receptor Regulatory Protein (TARP) γ-8.
Gardinier, Kevin M; Gernert, Douglas L; Porter, Warren J; Reel, Jon K; Ornstein, Paul L; Spinazze, Patrick; Stevens, F Craig; Hahn, Patric; Hollinshead, Sean P; Mayhugh, Daniel; Schkeryantz, Jeff; Khilevich, Albert; De Frutos, Oscar; Gleason, Scott D; Kato, Akihiko S; Luffer-Atlas, Debra; Desai, Prashant V; Swanson, Steven; Burris, Kevin D; Ding, Chunjin; Heinz, Beverly A; Need, Anne B; Barth, Vanessa N; Stephenson, Gregory A; Diseroad, Benjamin A; Woods, Tim A; Yu, Hong; Bredt, David; Witkin, Jeffrey M.
Afiliação
  • Gardinier KM; Lilly Research Laboratories, Eli Lilly and Company , Indianapolis, Indiana 46285 United States.
  • Gernert DL; Lilly Research Laboratories, Eli Lilly and Company , Indianapolis, Indiana 46285 United States.
  • Porter WJ; Lilly Research Laboratories, Eli Lilly and Company , Indianapolis, Indiana 46285 United States.
  • Reel JK; Lilly Research Laboratories, Eli Lilly and Company , Indianapolis, Indiana 46285 United States.
  • Ornstein PL; Lilly Research Laboratories, Eli Lilly and Company , Indianapolis, Indiana 46285 United States.
  • Spinazze P; Lilly Research Laboratories, Eli Lilly and Company , Indianapolis, Indiana 46285 United States.
  • Stevens FC; Lilly Research Laboratories, Eli Lilly and Company , Indianapolis, Indiana 46285 United States.
  • Hahn P; Lilly Research Laboratories, Eli Lilly and Company , Indianapolis, Indiana 46285 United States.
  • Hollinshead SP; Lilly Research Laboratories, Eli Lilly and Company , Indianapolis, Indiana 46285 United States.
  • Mayhugh D; Lilly Research Laboratories, Eli Lilly and Company , Indianapolis, Indiana 46285 United States.
  • Schkeryantz J; Lilly Research Laboratories, Eli Lilly and Company , Indianapolis, Indiana 46285 United States.
  • Khilevich A; Lilly Research Laboratories, Eli Lilly and Company , Indianapolis, Indiana 46285 United States.
  • De Frutos O; Lilly Research Laboratories, Eli Lilly and Company , Indianapolis, Indiana 46285 United States.
  • Gleason SD; Lilly Research Laboratories, Eli Lilly and Company , Indianapolis, Indiana 46285 United States.
  • Kato AS; Lilly Research Laboratories, Eli Lilly and Company , Indianapolis, Indiana 46285 United States.
  • Luffer-Atlas D; Lilly Research Laboratories, Eli Lilly and Company , Indianapolis, Indiana 46285 United States.
  • Desai PV; Lilly Research Laboratories, Eli Lilly and Company , Indianapolis, Indiana 46285 United States.
  • Swanson S; Lilly Research Laboratories, Eli Lilly and Company , Indianapolis, Indiana 46285 United States.
  • Burris KD; Lilly Research Laboratories, Eli Lilly and Company , Indianapolis, Indiana 46285 United States.
  • Ding C; Lilly Research Laboratories, Eli Lilly and Company , Indianapolis, Indiana 46285 United States.
  • Heinz BA; Lilly Research Laboratories, Eli Lilly and Company , Indianapolis, Indiana 46285 United States.
  • Need AB; Lilly Research Laboratories, Eli Lilly and Company , Indianapolis, Indiana 46285 United States.
  • Barth VN; Lilly Research Laboratories, Eli Lilly and Company , Indianapolis, Indiana 46285 United States.
  • Stephenson GA; Lilly Research Laboratories, Eli Lilly and Company , Indianapolis, Indiana 46285 United States.
  • Diseroad BA; Lilly Research Laboratories, Eli Lilly and Company , Indianapolis, Indiana 46285 United States.
  • Woods TA; Lilly Research Laboratories, Eli Lilly and Company , Indianapolis, Indiana 46285 United States.
  • Yu H; Lilly Research Laboratories, Eli Lilly and Company , Indianapolis, Indiana 46285 United States.
  • Bredt D; Lilly Research Laboratories, Eli Lilly and Company , Indianapolis, Indiana 46285 United States.
  • Witkin JM; Lilly Research Laboratories, Eli Lilly and Company , Indianapolis, Indiana 46285 United States.
J Med Chem ; 59(10): 4753-68, 2016 05 26.
Article em En | MEDLINE | ID: mdl-27067148

Texto completo: 1 Bases de dados: MEDLINE Assunto principal: Canais de Cálcio / Receptores de AMPA / Descoberta de Drogas Limite: Humans Idioma: En Revista: J Med Chem Assunto da revista: QUIMICA Ano de publicação: 2016 Tipo de documento: Article

Texto completo: 1 Bases de dados: MEDLINE Assunto principal: Canais de Cálcio / Receptores de AMPA / Descoberta de Drogas Limite: Humans Idioma: En Revista: J Med Chem Assunto da revista: QUIMICA Ano de publicação: 2016 Tipo de documento: Article