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Structure-activity relationship of uridine-based nucleoside phosphoramidate prodrugs for inhibition of dengue virus RNA-dependent RNA polymerase.
Wang, Gang; Lim, Siew Pheng; Chen, Yen-Liang; Hunziker, Jürg; Rao, Ranga; Gu, Feng; Seh, Cheah Chen; Ghafar, Nahdiyah Abdul; Xu, Haoying; Chan, Katherine; Lin, Xiaodong; Saunders, Oliver L; Fenaux, Martijn; Zhong, Weidong; Shi, Pei-Yong; Yokokawa, Fumiaki.
Afiliação
  • Wang G; Novartis Institute for Tropical Diseases, 10 Biopolis Road, #05-01 Chromos Singapore 138670, Singapore.
  • Lim SP; Novartis Institute for Tropical Diseases, 10 Biopolis Road, #05-01 Chromos Singapore 138670, Singapore.
  • Chen YL; Novartis Institute for Tropical Diseases, 10 Biopolis Road, #05-01 Chromos Singapore 138670, Singapore; Novartis Institutes for BioMedical Research, 5300 Chiron Way, Emeryville, CA 94608, United States.
  • Hunziker J; Novartis Institutes for BioMedical Research, Forum 1 Novartis Campus, CH-4056 Basel, Switzerland.
  • Rao R; Novartis Institute for Tropical Diseases, 10 Biopolis Road, #05-01 Chromos Singapore 138670, Singapore.
  • Gu F; Novartis Institute for Tropical Diseases, 10 Biopolis Road, #05-01 Chromos Singapore 138670, Singapore; Novartis Institutes for BioMedical Research, 5300 Chiron Way, Emeryville, CA 94608, United States.
  • Seh CC; Novartis Institute for Tropical Diseases, 10 Biopolis Road, #05-01 Chromos Singapore 138670, Singapore.
  • Ghafar NA; Novartis Institute for Tropical Diseases, 10 Biopolis Road, #05-01 Chromos Singapore 138670, Singapore.
  • Xu H; Novartis Institute for Tropical Diseases, 10 Biopolis Road, #05-01 Chromos Singapore 138670, Singapore.
  • Chan K; Novartis Institute for Tropical Diseases, 10 Biopolis Road, #05-01 Chromos Singapore 138670, Singapore; Novartis Institutes for BioMedical Research, 5300 Chiron Way, Emeryville, CA 94608, United States.
  • Lin X; Novartis Institutes for BioMedical Research, 5300 Chiron Way, Emeryville, CA 94608, United States.
  • Saunders OL; Novartis Institutes for BioMedical Research, 5300 Chiron Way, Emeryville, CA 94608, United States.
  • Fenaux M; Novartis Institutes for BioMedical Research, 5300 Chiron Way, Emeryville, CA 94608, United States.
  • Zhong W; Novartis Institutes for BioMedical Research, 5300 Chiron Way, Emeryville, CA 94608, United States.
  • Shi PY; Novartis Institute for Tropical Diseases, 10 Biopolis Road, #05-01 Chromos Singapore 138670, Singapore; Department of Biochemistry & Molecular Biology, Department of Pharmacology & Toxicology, Sealy Center for Structural Biology & Molecular Biophysics, University of Texas Medical Branch,
  • Yokokawa F; Novartis Institute for Tropical Diseases, 10 Biopolis Road, #05-01 Chromos Singapore 138670, Singapore; Novartis Institutes for BioMedical Research, 5300 Chiron Way, Emeryville, CA 94608, United States. Electronic address: fumiaki.yokokawa@novartis.com.
Bioorg Med Chem Lett ; 28(13): 2324-2327, 2018 07 15.
Article em En | MEDLINE | ID: mdl-29801997

Texto completo: 1 Bases de dados: MEDLINE Assunto principal: Antivirais / Uridina Monofosfato / RNA Polimerase Dependente de RNA / Pró-Fármacos / Inibidores Enzimáticos Limite: Humans Idioma: En Revista: Bioorg Med Chem Lett Assunto da revista: BIOQUIMICA / QUIMICA Ano de publicação: 2018 Tipo de documento: Article País de afiliação: Singapura

Texto completo: 1 Bases de dados: MEDLINE Assunto principal: Antivirais / Uridina Monofosfato / RNA Polimerase Dependente de RNA / Pró-Fármacos / Inibidores Enzimáticos Limite: Humans Idioma: En Revista: Bioorg Med Chem Lett Assunto da revista: BIOQUIMICA / QUIMICA Ano de publicação: 2018 Tipo de documento: Article País de afiliação: Singapura