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Discovery of 2-(1-(3-(4-Chloroxyphenyl)-3-oxo- propyl)pyrrolidine-3-yl)-1H-benzo[d]imidazole-4-carboxamide: A Potent Poly(ADP-ribose) Polymerase (PARP) Inhibitor for Treatment of Cancer.
Min, Rui; Wu, Weibin; Wang, Mingzhong; Tang, Lin; Chen, Dawei; Zhao, Huan; Zhang, Cunlong; Jiang, Yuyang.
Afiliação
  • Min R; Department of Chemistry, Tsinghua University, Beijing 100084, China. mr16@mails.tsinghua.edu.cn.
  • Wu W; The Ministry-Province Jointly Constructed Base for State Key Lab-Shenzhen Key Laboratory of Chemical Biology, The Graduate School at Shenzhen, Tsinghua University, Shenzhen 518055, China. mr16@mails.tsinghua.edu.cn.
  • Wang M; Shenzhen Kivita Innovative Drug Discovery Institute, Shenzhen 518055, China. weibin.wu@szkivita.com.
  • Tang L; Shenzhen Kivita Innovative Drug Discovery Institute, Shenzhen 518055, China. mzwang2000@163.com.
  • Chen D; Shenzhen Kivita Innovative Drug Discovery Institute, Shenzhen 518055, China. adamtl@126.com.
  • Zhao H; Shenzhen Kivita Innovative Drug Discovery Institute, Shenzhen 518055, China. dawei-ba@163.com.
  • Zhang C; Shenzhen Ruikang Pharmaceutical Technology Co. Ltd., Shenzhen 518055, China. zhaohuan8650@126.com.
  • Jiang Y; Shenzhen Kivita Innovative Drug Discovery Institute, Shenzhen 518055, China. zhcunl@126.com.
Molecules ; 24(10)2019 May 17.
Article em En | MEDLINE | ID: mdl-31108884

Texto completo: 1 Bases de dados: MEDLINE Assunto principal: Inibidores de Poli(ADP-Ribose) Polimerases / Imidazóis / Neoplasias Limite: Humans Idioma: En Revista: Molecules Assunto da revista: BIOLOGIA Ano de publicação: 2019 Tipo de documento: Article País de afiliação: China

Texto completo: 1 Bases de dados: MEDLINE Assunto principal: Inibidores de Poli(ADP-Ribose) Polimerases / Imidazóis / Neoplasias Limite: Humans Idioma: En Revista: Molecules Assunto da revista: BIOLOGIA Ano de publicação: 2019 Tipo de documento: Article País de afiliação: China