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Discovery of an Allosteric Ligand Binding Site in SMYD3 Lysine Methyltransferase.
Talibov, Vladimir O; Fabini, Edoardo; FitzGerald, Edward A; Tedesco, Daniele; Cederfeldt, Daniela; Talu, Martin J; Rachman, Moira M; Mihalic, Filip; Manoni, Elisabetta; Naldi, Marina; Sanese, Paola; Forte, Giovanna; Lepore Signorile, Martina; Barril, Xavier; Simone, Cristiano; Bartolini, Manuela; Dobritzsch, Doreen; Del Rio, Alberto; Danielson, U Helena.
Afiliação
  • Talibov VO; Department of Chemistry-BMC, Uppsala University, Husargatan 3, 754 24, Uppsala, Sweden.
  • Fabini E; Department of Pharmacy and Biotechnology, Alma Mater Studiorum University of Bologna, Via Belmeloro 6, 40126, Bologna, Italy.
  • FitzGerald EA; Institute for Organic Synthesis and Photoreactivity, National Research Council, Via P. Gobetti 101, 40129, Bologna, Italy.
  • Tedesco D; Department of Chemistry-BMC, Uppsala University, Husargatan 3, 754 24, Uppsala, Sweden.
  • Cederfeldt D; Beactica Therapeutics AB, Virdings allé 2, 754 50, Uppsala, Sweden.
  • Talu MJ; Department of Pharmacy and Biotechnology, Alma Mater Studiorum University of Bologna, Via Belmeloro 6, 40126, Bologna, Italy.
  • Rachman MM; Institute for Organic Synthesis and Photoreactivity, National Research Council, Via P. Gobetti 101, 40129, Bologna, Italy.
  • Mihalic F; Department of Chemistry-BMC, Uppsala University, Husargatan 3, 754 24, Uppsala, Sweden.
  • Manoni E; Department of Chemistry-BMC, Uppsala University, Husargatan 3, 754 24, Uppsala, Sweden.
  • Naldi M; Institut de Biomedicina de la Universitat de Barcelona (IBUB) and Facultat de Farmacia, Universitat de Barcelona, Av. Joan XXIII 27-31, 08028, Barcelona, Spain.
  • Sanese P; Department of Chemistry-BMC, Uppsala University, Husargatan 3, 754 24, Uppsala, Sweden.
  • Forte G; Institute for Organic Synthesis and Photoreactivity, National Research Council, Via P. Gobetti 101, 40129, Bologna, Italy.
  • Lepore Signorile M; Department of Pharmacy and Biotechnology, Alma Mater Studiorum University of Bologna, Via Belmeloro 6, 40126, Bologna, Italy.
  • Barril X; Centre for Applied Biomedical Research, Alma Mater Studiorum University of Bologna, Via Zamboni, 33, Bologna, 40126, Italy.
  • Simone C; Medical Genetics, National Institute for Gastroenterology, IRCCS 'S. de Bellis' Research Hospital, 70013, Bari, Italy.
  • Bartolini M; Medical Genetics, National Institute for Gastroenterology, IRCCS 'S. de Bellis' Research Hospital, 70013, Bari, Italy.
  • Dobritzsch D; Medical Genetics, National Institute for Gastroenterology, IRCCS 'S. de Bellis' Research Hospital, 70013, Bari, Italy.
  • Del Rio A; Institut de Biomedicina de la Universitat de Barcelona (IBUB) and Facultat de Farmacia, Universitat de Barcelona, Av. Joan XXIII 27-31, 08028, Barcelona, Spain.
  • Danielson UH; Catalan Institution for Research and Advanced Studies (ICREA), Passeig Lluis Companys 23, 08010, Barcelona, Spain.
Chembiochem ; 22(9): 1597-1608, 2021 05 04.
Article em En | MEDLINE | ID: mdl-33400854

Texto completo: 1 Bases de dados: MEDLINE Assunto principal: Histona-Lisina N-Metiltransferase / Proteínas de Choque Térmico HSP90 Limite: Humans Idioma: En Revista: Chembiochem Assunto da revista: BIOQUIMICA Ano de publicação: 2021 Tipo de documento: Article País de afiliação: Suécia

Texto completo: 1 Bases de dados: MEDLINE Assunto principal: Histona-Lisina N-Metiltransferase / Proteínas de Choque Térmico HSP90 Limite: Humans Idioma: En Revista: Chembiochem Assunto da revista: BIOQUIMICA Ano de publicação: 2021 Tipo de documento: Article País de afiliação: Suécia