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Development of 18F-Labeled Radiotracers for PET Imaging of the Adenosine A2A Receptor: Synthesis, Radiolabeling and Preliminary Biological Evaluation.
Lai, Thu Hang; Schröder, Susann; Toussaint, Magali; Dukic-Stefanovic, Sladjana; Kranz, Mathias; Ludwig, Friedrich-Alexander; Fischer, Steffen; Steinbach, Jörg; Deuther-Conrad, Winnie; Brust, Peter; Moldovan, Rares-Petru.
Afiliação
  • Lai TH; Helmholtz-Zentrum Dresden-Rossendorf (HZDR), Department of Neuroradiopharmaceuticals, Institute of Radiopharmaceutical Cancer Research, Research site Leipzig, 04318 Leipzig, Germany.
  • Schröder S; Department of Research and Development, ROTOP Pharmaka Ltd., Dresden 01328, Germany.
  • Toussaint M; Department of Research and Development, ROTOP Pharmaka Ltd., Dresden 01328, Germany.
  • Dukic-Stefanovic S; Helmholtz-Zentrum Dresden-Rossendorf (HZDR), Department of Neuroradiopharmaceuticals, Institute of Radiopharmaceutical Cancer Research, Research site Leipzig, 04318 Leipzig, Germany.
  • Kranz M; Helmholtz-Zentrum Dresden-Rossendorf (HZDR), Department of Neuroradiopharmaceuticals, Institute of Radiopharmaceutical Cancer Research, Research site Leipzig, 04318 Leipzig, Germany.
  • Ludwig FA; Helmholtz-Zentrum Dresden-Rossendorf (HZDR), Department of Neuroradiopharmaceuticals, Institute of Radiopharmaceutical Cancer Research, Research site Leipzig, 04318 Leipzig, Germany.
  • Fischer S; PET Imaging Center, University Hospital of North Norway (UNN), 9009 Tromsø, Norway.
  • Steinbach J; Nuclear Medicine and Radiation Biology Research Group, The Arctic University of Norway, 9009 Tromsø, Norway.
  • Deuther-Conrad W; Helmholtz-Zentrum Dresden-Rossendorf (HZDR), Department of Neuroradiopharmaceuticals, Institute of Radiopharmaceutical Cancer Research, Research site Leipzig, 04318 Leipzig, Germany.
  • Brust P; Helmholtz-Zentrum Dresden-Rossendorf (HZDR), Department of Neuroradiopharmaceuticals, Institute of Radiopharmaceutical Cancer Research, Research site Leipzig, 04318 Leipzig, Germany.
  • Moldovan RP; Helmholtz-Zentrum Dresden-Rossendorf (HZDR), Department of Neuroradiopharmaceuticals, Institute of Radiopharmaceutical Cancer Research, Research site Leipzig, 04318 Leipzig, Germany.
Int J Mol Sci ; 22(5)2021 Feb 25.
Article em En | MEDLINE | ID: mdl-33669003

Texto completo: 1 Bases de dados: MEDLINE Assunto principal: Encéfalo / Radioisótopos de Flúor / Compostos Radiofarmacêuticos / Receptor A2A de Adenosina / Tomografia por Emissão de Pósitrons / Hidrocarbonetos Fluorados Limite: Animals Idioma: En Revista: Int J Mol Sci Ano de publicação: 2021 Tipo de documento: Article País de afiliação: Alemanha

Texto completo: 1 Bases de dados: MEDLINE Assunto principal: Encéfalo / Radioisótopos de Flúor / Compostos Radiofarmacêuticos / Receptor A2A de Adenosina / Tomografia por Emissão de Pósitrons / Hidrocarbonetos Fluorados Limite: Animals Idioma: En Revista: Int J Mol Sci Ano de publicação: 2021 Tipo de documento: Article País de afiliação: Alemanha