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A Solid Supported Membrane-Based Technology for Electrophysical Screening of B0AT1-Modulating Compounds.
Gerbeth-Kreul, Carolin; Pommereau, Antje; Ruf, Sven; Kane, John L; Kuntzweiler, Theresa; Hessler, Gerhard; Engel, Christian K; Shum, Patrick; Wei, LinLi; Czech, Joerg; Licher, Thomas.
Afiliação
  • Gerbeth-Kreul C; In Vitro Biology & High-throughput Chemistry, Integrated Drug Discovery, Sanofi-Aventis Deutschland GmbH, Frankfurt, Germany.
  • Pommereau A; In Vitro Biology & High-throughput Chemistry, Integrated Drug Discovery, Sanofi-Aventis Deutschland GmbH, Frankfurt, Germany.
  • Ruf S; Synthetic Molecular Design, Integrated Drug Discovery, Sanofi-Aventis Deutschland GmbH, Frankfurt, Germany.
  • Kane JL; Medicinal Chemistry, Integrated Drug Discovery, Sanofi-Genzyme, Waltham, MA, USA.
  • Kuntzweiler T; In Vitro Biology, Integrated Drug Discovery, Sanofi-Genzyme, Waltham, MA, USA.
  • Hessler G; Synthetic Molecular Design, Integrated Drug Discovery, Sanofi-Aventis Deutschland GmbH, Frankfurt, Germany.
  • Engel CK; Synthetic Molecular Design, Integrated Drug Discovery, Sanofi-Aventis Deutschland GmbH, Frankfurt, Germany.
  • Shum P; Medicinal Chemistry, Integrated Drug Discovery, Sanofi-Genzyme, Waltham, MA, USA.
  • Wei L; Medicinal Chemistry, Integrated Drug Discovery, Sanofi-Genzyme, Waltham, MA, USA.
  • Czech J; In Vitro Biology & High-throughput Chemistry, Integrated Drug Discovery, Sanofi-Aventis Deutschland GmbH, Frankfurt, Germany.
  • Licher T; In Vitro Biology & High-throughput Chemistry, Integrated Drug Discovery, Sanofi-Aventis Deutschland GmbH, Frankfurt, Germany.
SLAS Discov ; 26(6): 783-797, 2021 07.
Article em En | MEDLINE | ID: mdl-33955247

Texto completo: 1 Bases de dados: MEDLINE Assunto principal: Sistemas de Transporte de Aminoácidos Neutros / Fenômenos Eletrofisiológicos / Ensaios de Triagem em Larga Escala Tipo de estudo: Diagnostic_studies / Evaluation_studies / Prognostic_studies / Screening_studies Limite: Animals / Humans Idioma: En Revista: SLAS Discov Ano de publicação: 2021 Tipo de documento: Article País de afiliação: Alemanha

Texto completo: 1 Bases de dados: MEDLINE Assunto principal: Sistemas de Transporte de Aminoácidos Neutros / Fenômenos Eletrofisiológicos / Ensaios de Triagem em Larga Escala Tipo de estudo: Diagnostic_studies / Evaluation_studies / Prognostic_studies / Screening_studies Limite: Animals / Humans Idioma: En Revista: SLAS Discov Ano de publicação: 2021 Tipo de documento: Article País de afiliação: Alemanha