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Identification and characterization of two drug-like fragments that bind to the same cryptic binding pocket of Burkholderia pseudomallei DsbA.
Petit, Guillaume A; Mohanty, Biswaranjan; McMahon, Róisín M; Nebl, Stefan; Hilko, David H; Wilde, Karyn L; Scanlon, Martin J; Martin, Jennifer L; Halili, Maria A.
Afiliação
  • Petit GA; Griffith Institute for Drug Discovery, Griffith University, Building N75, 46 Don Young Road, Nathan, QLD 4111, Australia.
  • Mohanty B; Medicinal Chemistry, Monash Institute of Pharmaceutical Sciences, Monash University, 381 Royal Parade, Parkville, VIC 3052, Australia.
  • McMahon RM; Griffith Institute for Drug Discovery, Griffith University, Building N75, 46 Don Young Road, Nathan, QLD 4111, Australia.
  • Nebl S; Medicinal Chemistry, Monash Institute of Pharmaceutical Sciences, Monash University, 381 Royal Parade, Parkville, VIC 3052, Australia.
  • Hilko DH; Griffith Institute for Drug Discovery, Griffith University, Building N75, 46 Don Young Road, Nathan, QLD 4111, Australia.
  • Wilde KL; National Deuteration Facility, Australian Nuclear Science and Technology Organization (ANSTO), New Illawarra Road, Lucas Heights, NSW 2234, Australia.
  • Scanlon MJ; Medicinal Chemistry, Monash Institute of Pharmaceutical Sciences, Monash University, 381 Royal Parade, Parkville, VIC 3052, Australia.
  • Martin JL; Griffith Institute for Drug Discovery, Griffith University, Building N75, 46 Don Young Road, Nathan, QLD 4111, Australia.
  • Halili MA; Griffith Institute for Drug Discovery, Griffith University, Building N75, 46 Don Young Road, Nathan, QLD 4111, Australia.
Acta Crystallogr D Struct Biol ; 78(Pt 1): 75-90, 2022 Jan 01.
Article em En | MEDLINE | ID: mdl-34981764

Texto completo: 1 Bases de dados: MEDLINE Assunto principal: Burkholderia pseudomallei / Antibacterianos Tipo de estudo: Diagnostic_studies / Prognostic_studies Idioma: En Revista: Acta Crystallogr D Struct Biol Ano de publicação: 2022 Tipo de documento: Article País de afiliação: Austrália

Texto completo: 1 Bases de dados: MEDLINE Assunto principal: Burkholderia pseudomallei / Antibacterianos Tipo de estudo: Diagnostic_studies / Prognostic_studies Idioma: En Revista: Acta Crystallogr D Struct Biol Ano de publicação: 2022 Tipo de documento: Article País de afiliação: Austrália