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Design, synthesis, SAR, and biological evaluation of saccharin-based hybrids as carbonic anhydrase inhibitors.
Chinchilli, Krishna K; Royyala, Venkata N; Thacker, Pavitra S; Angeli, Andrea; Danaboina, Srikanth; Singh, Priti; Nanduri, Srinivas; Supuran, Claudiu T; Arifuddin, Mohammed.
Afiliação
  • Chinchilli KK; Department of Medicinal Chemistry, National Institute of Pharmaceutical Education and Research (NIPER), Hyderabad, India.
  • Royyala VN; Department of Medicinal Chemistry, National Institute of Pharmaceutical Education and Research (NIPER), Hyderabad, India.
  • Thacker PS; Department of Medicinal Chemistry, National Institute of Pharmaceutical Education and Research (NIPER), Hyderabad, India.
  • Angeli A; Neurofarba Department, Sezione di Scienze, Farmaceutiche e Nutraceutiche, Università Degli Studi di Firenze, Florence, Italy.
  • Danaboina S; Department of Medicinal Chemistry, National Institute of Pharmaceutical Education and Research (NIPER), Hyderabad, India.
  • Singh P; Process Chemistry Process Technology, Department of Chemical Sciences, National Institute of Pharmaceutical Education and Research (NIPER), Hyderabad, India.
  • Nanduri S; Process Chemistry Process Technology, Department of Chemical Sciences, National Institute of Pharmaceutical Education and Research (NIPER), Hyderabad, India.
  • Supuran CT; Neurofarba Department, Sezione di Scienze, Farmaceutiche e Nutraceutiche, Università Degli Studi di Firenze, Florence, Italy.
  • Arifuddin M; Department of Medicinal Chemistry, National Institute of Pharmaceutical Education and Research (NIPER), Hyderabad, India.
Arch Pharm (Weinheim) ; 355(8): e2200019, 2022 Aug.
Article em En | MEDLINE | ID: mdl-35484599

Texto completo: 1 Bases de dados: MEDLINE Assunto principal: Inibidores da Anidrase Carbônica / Anidrases Carbônicas Limite: Humans Idioma: En Revista: Arch Pharm (Weinheim) Ano de publicação: 2022 Tipo de documento: Article País de afiliação: Índia

Texto completo: 1 Bases de dados: MEDLINE Assunto principal: Inibidores da Anidrase Carbônica / Anidrases Carbônicas Limite: Humans Idioma: En Revista: Arch Pharm (Weinheim) Ano de publicação: 2022 Tipo de documento: Article País de afiliação: Índia