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Discovery of pyrazole-1-carboxamide derivatives as novel Gi-biased µ-opioid receptor agonists.
Jung, Jae-Hoon; Jang, In Hee; Kim, Yeo Ok; Kim, Sunhong; Yoon, Myung Ha; Kim, Yong-Chul.
Afiliação
  • Jung JH; School of Life Sciences, Gwangju Institute of Science and Technology (GIST), Gwangju, Republic of Korea.
  • Jang IH; Disease Target Structure Research Center, Korea Research Institute of Bioscience and Biotechnology, Daejeon, Republic of Korea.
  • Kim YO; College of Pharmacy, Chungnam National University, Daejeon, Republic of Korea.
  • Kim S; Department of Anesthesiology and Pain Medicine, Medical School, Chonnam National University, Gwangju, Republic of Korea.
  • Yoon MH; Disease Target Structure Research Center, Korea Research Institute of Bioscience and Biotechnology, Daejeon, Republic of Korea.
  • Kim YC; Department of Biomolecular Science, KRIBB School of Biological Science, Korea University of Science and Technology, Daejeon, Republic of Korea.
Drug Dev Res ; 83(7): 1600-1612, 2022 11.
Article em En | MEDLINE | ID: mdl-36124859

Texto completo: 1 Bases de dados: MEDLINE Assunto principal: Receptores Opioides mu / Neuralgia Limite: Humans Idioma: En Revista: Drug Dev Res Ano de publicação: 2022 Tipo de documento: Article

Texto completo: 1 Bases de dados: MEDLINE Assunto principal: Receptores Opioides mu / Neuralgia Limite: Humans Idioma: En Revista: Drug Dev Res Ano de publicação: 2022 Tipo de documento: Article