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Silmitasertib (CX-4945), a Clinically Used CK2-Kinase Inhibitor with Additional Effects on GSK3ß and DYRK1A Kinases: A Structural Perspective.
Grygier, Przemyslaw; Pustelny, Katarzyna; Nowak, Jakub; Golik, Przemyslaw; Popowicz, Grzegorz M; Plettenburg, Oliver; Dubin, Grzegorz; Menezes, Filipe; Czarna, Anna.
Afiliação
  • Grygier P; Malopolska Centre of Biotechnology, Jagiellonian University, Gronostajowa 7A, 30-387 Krakow, Poland.
  • Pustelny K; Malopolska Centre of Biotechnology, Jagiellonian University, Gronostajowa 7A, 30-387 Krakow, Poland.
  • Nowak J; Malopolska Centre of Biotechnology, Jagiellonian University, Gronostajowa 7A, 30-387 Krakow, Poland.
  • Golik P; Selvita S.A, Bobrzynskiego, 14, 30-338 Krakow, Poland.
  • Popowicz GM; Institute of Structural Biology, Helmholtz Zentrum Muenchen, Ingolstaedter Landstrasse 1, Neuherberg 85764, Germany.
  • Plettenburg O; Biomolecular NMR and Center for Integrated Protein Science Munich at Department Chemie, Technical University of Munich, Lichtenbergstrasse 4, Garching 85747, Germany.
  • Dubin G; Institute of Medicinal Chemistry, Helmholtz Munich, Ingolstaedter Landstrasse 1, Neuherberg 85764, Germany.
  • Menezes F; Institute of Organic Chemistry, Centre of Biomolecular Drug Research (BMWZ) and Laboratory of Nano and Quantum Engineering (LNQE), Leibniz University Hannover, Schneiderberg 1b, Hannover 30167, Germany.
  • Czarna A; German Center for Diabetes Research (DZD), Ingolstaedter Landstrasse 1, Neuherberg 85764, Germany.
J Med Chem ; 66(6): 4009-4024, 2023 03 23.
Article em En | MEDLINE | ID: mdl-36883902

Texto completo: 1 Bases de dados: MEDLINE Assunto principal: Caseína Quinase II / Naftiridinas Idioma: En Revista: J Med Chem Assunto da revista: QUIMICA Ano de publicação: 2023 Tipo de documento: Article País de afiliação: Polônia

Texto completo: 1 Bases de dados: MEDLINE Assunto principal: Caseína Quinase II / Naftiridinas Idioma: En Revista: J Med Chem Assunto da revista: QUIMICA Ano de publicação: 2023 Tipo de documento: Article País de afiliação: Polônia