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Development of Masitinib Derivatives with Enhanced Mpro Ligand Efficiency and Reduced Cytotoxicity.
Menendez, Cintia A; Mohamed, Adil; Perez-Lemus, Gustavo R; Weiss, Adam M; Rawe, Benjamin W; Liu, Guancen; Crolais, Alex E; Kenna, Emma; Byléhn, Fabian; Alvarado, Walter; Mendels, Dan; Rowan, Stuart J; Tay, Savas; de Pablo, Juan J.
Afiliação
  • Menendez CA; Pritzker School of Molecular Engineering, University of Chicago, 5640 South Ellis Avenue, Chicago, IL 60637, USA.
  • Mohamed A; Pritzker School of Molecular Engineering, University of Chicago, 5640 South Ellis Avenue, Chicago, IL 60637, USA.
  • Perez-Lemus GR; Pritzker School of Molecular Engineering, University of Chicago, 5640 South Ellis Avenue, Chicago, IL 60637, USA.
  • Weiss AM; Department of Chemistry, University of Chicago, 5735 South Ellis Avenue, Chicago, IL 60637, USA.
  • Rawe BW; Pritzker School of Molecular Engineering, University of Chicago, 5640 South Ellis Avenue, Chicago, IL 60637, USA.
  • Liu G; Department of Chemistry, University of Chicago, 5735 South Ellis Avenue, Chicago, IL 60637, USA.
  • Crolais AE; Department of Chemistry, University of Chicago, 5735 South Ellis Avenue, Chicago, IL 60637, USA.
  • Kenna E; Pritzker School of Molecular Engineering, University of Chicago, 5640 South Ellis Avenue, Chicago, IL 60637, USA.
  • Byléhn F; Pritzker School of Molecular Engineering, University of Chicago, 5640 South Ellis Avenue, Chicago, IL 60637, USA.
  • Alvarado W; Pritzker School of Molecular Engineering, University of Chicago, 5640 South Ellis Avenue, Chicago, IL 60637, USA.
  • Mendels D; Pritzker School of Molecular Engineering, University of Chicago, 5640 South Ellis Avenue, Chicago, IL 60637, USA.
  • Rowan SJ; Pritzker School of Molecular Engineering, University of Chicago, 5640 South Ellis Avenue, Chicago, IL 60637, USA.
  • Tay S; Department of Chemistry, University of Chicago, 5735 South Ellis Avenue, Chicago, IL 60637, USA.
  • de Pablo JJ; Pritzker School of Molecular Engineering, University of Chicago, 5640 South Ellis Avenue, Chicago, IL 60637, USA.
Molecules ; 28(18)2023 Sep 15.
Article em En | MEDLINE | ID: mdl-37764425

Texto completo: 1 Bases de dados: MEDLINE Assunto principal: Piperidinas / Piridinas / Benzamidas Limite: Humans Idioma: En Revista: Molecules Assunto da revista: BIOLOGIA Ano de publicação: 2023 Tipo de documento: Article País de afiliação: Estados Unidos

Texto completo: 1 Bases de dados: MEDLINE Assunto principal: Piperidinas / Piridinas / Benzamidas Limite: Humans Idioma: En Revista: Molecules Assunto da revista: BIOLOGIA Ano de publicação: 2023 Tipo de documento: Article País de afiliação: Estados Unidos