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Benzimidazole derivatives as tubulin polymerization inhibitors: Design, synthesis and in vitro cytotoxicity studies.
Laxmikeshav, Kritika; Rahman, Ziaur; Mahale, Ashutosh; Gurukkala Valapil, Durgesh; Sharma, Pravesh; George, Joel; Phanindranath, Regur; Dandekar, Manoj P; Kulkarni, Onkar P; Nagesh, Narayana; Shankaraiah, Nagula.
Afiliação
  • Laxmikeshav K; Department of Medicinal Chemistry, National Institute of Pharmaceutical Education and Research (NIPER), Hyderabad 500037, India.
  • Rahman Z; Department of Biological Sciences, National Institute of Pharmaceutical Education and Research (NIPER), Hyderabad 500037, India.
  • Mahale A; Department of Pharmacy, Birla Institute of Technology and Science-Pilani, Hyderabad Campus, Hyderabad 500078, India.
  • Gurukkala Valapil D; Department of Medicinal Chemistry, National Institute of Pharmaceutical Education and Research (NIPER), Hyderabad 500037, India.
  • Sharma P; Department of Pharmacy, Birla Institute of Technology and Science-Pilani, Hyderabad Campus, Hyderabad 500078, India.
  • George J; CSIR-Centre for Cellular and Molecular Biology, Medical Biotechnology Complex, ANNEXE II, Uppal Road, Hyderabad 500007, India.
  • Phanindranath R; CSIR-Centre for Cellular and Molecular Biology, Medical Biotechnology Complex, ANNEXE II, Uppal Road, Hyderabad 500007, India.
  • Dandekar MP; Department of Biological Sciences, National Institute of Pharmaceutical Education and Research (NIPER), Hyderabad 500037, India. Electronic address: manoj.dandekar@niperhyd.ac.in.
  • Kulkarni OP; Department of Pharmacy, Birla Institute of Technology and Science-Pilani, Hyderabad Campus, Hyderabad 500078, India.
  • Nagesh N; CSIR-Centre for Cellular and Molecular Biology, Medical Biotechnology Complex, ANNEXE II, Uppal Road, Hyderabad 500007, India.
  • Shankaraiah N; Department of Medicinal Chemistry, National Institute of Pharmaceutical Education and Research (NIPER), Hyderabad 500037, India. Electronic address: shankar@niperhyd.ac.in.
Bioorg Med Chem Lett ; 96: 129494, 2023 11 15.
Article em En | MEDLINE | ID: mdl-37797804

Texto completo: 1 Bases de dados: MEDLINE Assunto principal: Moduladores de Tubulina / Antineoplásicos Limite: Animals / Humans Idioma: En Revista: Bioorg Med Chem Lett Assunto da revista: BIOQUIMICA / QUIMICA Ano de publicação: 2023 Tipo de documento: Article País de afiliação: Índia

Texto completo: 1 Bases de dados: MEDLINE Assunto principal: Moduladores de Tubulina / Antineoplásicos Limite: Animals / Humans Idioma: En Revista: Bioorg Med Chem Lett Assunto da revista: BIOQUIMICA / QUIMICA Ano de publicação: 2023 Tipo de documento: Article País de afiliação: Índia