Detalhe da pesquisa
1.
1,2,4-Triazole-3-thione analogues with an arylakyl group at position 4 as metallo-ß-lactamase inhibitors.
Bioorg Med Chem
; 72: 116964, 2022 10 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-36030663
2.
4-Alkyl-1,2,4-triazole-3-thione analogues as metallo-ß-lactamase inhibitors.
Bioorg Chem
; 113: 105024, 2021 08.
Artigo
em Inglês
| MEDLINE | ID: mdl-34116340
3.
Insights from structure-activity relationships and the binding mode of peptidic α-ketoamide inhibitors of the malaria drug target subtilisin-like SUB1.
Eur J Med Chem
; 269: 116308, 2024 Apr 05.
Artigo
em Inglês
| MEDLINE | ID: mdl-38503166
4.
1,2,4-Triazole-3-Thione Analogues with a 2-Ethylbenzoic Acid at Position 4 as VIM-type Metallo-ß-Lactamase Inhibitors.
ChemMedChem
; 17(7): e202100699, 2022 04 05.
Artigo
em Inglês
| MEDLINE | ID: mdl-35050549
5.
Optimization of 1,2,4-Triazole-3-thiones toward Broad-Spectrum Metallo-ß-lactamase Inhibitors Showing Potent Synergistic Activity on VIM- and NDM-1-Producing Clinical Isolates.
J Med Chem
; 65(24): 16392-16419, 2022 12 22.
Artigo
em Inglês
| MEDLINE | ID: mdl-36450011
6.
1,2,4-Triazole-3-thione compounds with a 4-ethyl alkyl/aryl sulfide substituent are broad-spectrum metallo-ß-lactamase inhibitors with re-sensitization activity.
Eur J Med Chem
; 226: 113873, 2021 Dec 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-34626878
7.
4-(N-Alkyl- and -Acyl-amino)-1,2,4-triazole-3-thione Analogs as Metallo-ß-Lactamase Inhibitors: Impact of 4-Linker on Potency and Spectrum of Inhibition.
Biomolecules
; 10(8)2020 07 23.
Artigo
em Inglês
| MEDLINE | ID: mdl-32717907
8.
4-Amino-1,2,4-triazole-3-thione-derived Schiff bases as metallo-ß-lactamase inhibitors.
Eur J Med Chem
; 208: 112720, 2020 Dec 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-32937203