1.
Bioorg Med Chem Lett
; 17(5): 1392-8, 2007 Mar 01.
Artigo
em Inglês
| MEDLINE
| ID: mdl-17194584
RESUMO
A 1,6-naphthyridine inhibitor of HIV-1 integrase has been discovered with excellent inhibitory activity in cells, good pharmacokinetics, and an excellent ability to inhibit virus with mutant enzyme.