Detalhe da pesquisa
1.
The potent and selective RIPK2 inhibitor BI 706039 improves intestinal inflammation in the TRUC mouse model of inflammatory bowel disease.
Am J Physiol Gastrointest Liver Physiol
; 321(5): G500-G512, 2021 11 01.
Artigo
em Inglês
| MEDLINE | ID: mdl-34494462
2.
Structural studies unravel the active conformation of apo RORγt nuclear receptor and a common inverse agonism of two diverse classes of RORγt inhibitors.
J Biol Chem
; 292(28): 11618-11630, 2017 07 14.
Artigo
em Inglês
| MEDLINE | ID: mdl-28546429
3.
Discovery of a Series of Pyrazinone RORγ Antagonists and Identification of the Clinical Candidate BI 730357.
ACS Med Chem Lett
; 12(1): 143-154, 2021 Jan 14.
Artigo
em Inglês
| MEDLINE | ID: mdl-33488976
4.
Discovery and SAR study of novel dihydroquinoline-containing glucocorticoid receptor agonists.
Bioorg Med Chem Lett
; 17(18): 5091-5, 2007 Sep 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-17681466
5.
Discovery and SAR study of novel dihydroquinoline containing glucocorticoid receptor ligands.
Bioorg Med Chem Lett
; 16(6): 1549-52, 2006 Mar 15.
Artigo
em Inglês
| MEDLINE | ID: mdl-16386422