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Discovery of a Potent, S1P3-Sparing Benzothiazole Agonist of Sphingosine-1-Phosphate Receptor 1 (S1P1).
Lanman, Brian A; Cee, Victor J; Cheruku, Srinivasa R; Frohn, Mike; Golden, Jennifer; Lin, Jian; Lobera, Mercedes; Marantz, Yael; Muller, Kristine M; Neira, Susana C; Pickrell, Alexander J; Rivenzon-Segal, Dalia; Schutz, Nili; Sharadendu, Anurag; Yu, Xiang; Zhang, Zhaoda; Buys, Janet; Fiorino, Mike; Gore, Anu; Horner, Michelle; Itano, Andrea; McElvain, Michele; Middleton, Scot; Schrag, Michael; Vargas, Hugo M; Xu, Han; Xu, Yang; Zhang, Xuxia; Siu, Jerry; Bürli, Roland W.
Afiliação
  • Lanman BA; Amgen Inc., One Amgen Center Drive, Thousand Oaks, California 91320, United States.
  • Cee VJ; Amgen Inc., One Amgen Center Drive, Thousand Oaks, California 91320, United States.
  • Cheruku SR; EPIX Pharmaceuticals Inc., 167 Worcester Street, Suite 201, Wellesley Hills, Massachusetts 02481, United States.
  • Frohn M; Amgen Inc., One Amgen Center Drive, Thousand Oaks, California 91320, United States.
  • Golden J; Amgen Inc., One Amgen Center Drive, Thousand Oaks, California 91320, United States.
  • Lin J; EPIX Pharmaceuticals Inc., 167 Worcester Street, Suite 201, Wellesley Hills, Massachusetts 02481, United States.
  • Lobera M; EPIX Pharmaceuticals Inc., 167 Worcester Street, Suite 201, Wellesley Hills, Massachusetts 02481, United States.
  • Marantz Y; EPIX Pharmaceuticals Inc., 167 Worcester Street, Suite 201, Wellesley Hills, Massachusetts 02481, United States.
  • Muller KM; Amgen Inc., One Amgen Center Drive, Thousand Oaks, California 91320, United States.
  • Neira SC; Amgen Inc., One Amgen Center Drive, Thousand Oaks, California 91320, United States.
  • Pickrell AJ; Amgen Inc., One Amgen Center Drive, Thousand Oaks, California 91320, United States.
  • Rivenzon-Segal D; EPIX Pharmaceuticals Inc., 167 Worcester Street, Suite 201, Wellesley Hills, Massachusetts 02481, United States.
  • Schutz N; EPIX Pharmaceuticals Inc., 167 Worcester Street, Suite 201, Wellesley Hills, Massachusetts 02481, United States.
  • Sharadendu A; EPIX Pharmaceuticals Inc., 167 Worcester Street, Suite 201, Wellesley Hills, Massachusetts 02481, United States.
  • Yu X; EPIX Pharmaceuticals Inc., 167 Worcester Street, Suite 201, Wellesley Hills, Massachusetts 02481, United States.
  • Zhang Z; EPIX Pharmaceuticals Inc., 167 Worcester Street, Suite 201, Wellesley Hills, Massachusetts 02481, United States.
  • Buys J; Amgen Inc., One Amgen Center Drive, Thousand Oaks, California 91320, United States.
  • Fiorino M; Amgen Inc., One Amgen Center Drive, Thousand Oaks, California 91320, United States.
  • Gore A; Amgen Inc., One Amgen Center Drive, Thousand Oaks, California 91320, United States.
  • Horner M; Amgen Inc., One Amgen Center Drive, Thousand Oaks, California 91320, United States.
  • Itano A; Amgen Inc., One Amgen Center Drive, Thousand Oaks, California 91320, United States.
  • McElvain M; Amgen Inc., One Amgen Center Drive, Thousand Oaks, California 91320, United States.
  • Middleton S; Amgen Inc., One Amgen Center Drive, Thousand Oaks, California 91320, United States.
  • Schrag M; Amgen Inc., One Amgen Center Drive, Thousand Oaks, California 91320, United States.
  • Vargas HM; Amgen Inc., One Amgen Center Drive, Thousand Oaks, California 91320, United States.
  • Xu H; Amgen Inc., One Amgen Center Drive, Thousand Oaks, California 91320, United States.
  • Xu Y; Amgen Inc., One Amgen Center Drive, Thousand Oaks, California 91320, United States.
  • Zhang X; Amgen Inc., One Amgen Center Drive, Thousand Oaks, California 91320, United States.
  • Siu J; Amgen Inc., One Amgen Center Drive, Thousand Oaks, California 91320, United States.
  • Bürli RW; Amgen Inc., One Amgen Center Drive, Thousand Oaks, California 91320, United States.
ACS Med Chem Lett ; 2(2): 102-6, 2011 Feb 10.
Article em En | MEDLINE | ID: mdl-24900287

Texto completo: 1 Base de dados: MEDLINE Idioma: En Ano de publicação: 2011 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Idioma: En Ano de publicação: 2011 Tipo de documento: Article