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Discovery of novel AKT inhibitors with enhanced anti-tumor effects in combination with the MEK inhibitor.
Dumble, Melissa; Crouthamel, Ming-Chih; Zhang, Shu-Yun; Schaber, Michael; Levy, Dana; Robell, Kimberly; Liu, Qi; Figueroa, David J; Minthorn, Elisabeth A; Seefeld, Mark A; Rouse, Meagan B; Rabindran, Sridhar K; Heerding, Dirk A; Kumar, Rakesh.
Afiliação
  • Dumble M; Oncology R & D, GlaxoSmithKline, Collegeville, Pennsylvania, United States of America.
  • Crouthamel MC; Oncology R & D, GlaxoSmithKline, Collegeville, Pennsylvania, United States of America.
  • Zhang SY; Oncology R & D, GlaxoSmithKline, Collegeville, Pennsylvania, United States of America.
  • Schaber M; Platform Technology & Science, GlaxoSmithKline, Collegeville, Pennsylvania, United States of America.
  • Levy D; Oncology R & D, GlaxoSmithKline, Collegeville, Pennsylvania, United States of America.
  • Robell K; Oncology R & D, GlaxoSmithKline, Collegeville, Pennsylvania, United States of America.
  • Liu Q; Oncology R & D, GlaxoSmithKline, Collegeville, Pennsylvania, United States of America.
  • Figueroa DJ; Oncology R & D, GlaxoSmithKline, Collegeville, Pennsylvania, United States of America.
  • Minthorn EA; Oncology R & D, GlaxoSmithKline, Collegeville, Pennsylvania, United States of America.
  • Seefeld MA; Oncology R & D, GlaxoSmithKline, Collegeville, Pennsylvania, United States of America.
  • Rouse MB; Oncology R & D, GlaxoSmithKline, Collegeville, Pennsylvania, United States of America.
  • Rabindran SK; Oncology R & D, GlaxoSmithKline, Collegeville, Pennsylvania, United States of America.
  • Heerding DA; Oncology R & D, GlaxoSmithKline, Collegeville, Pennsylvania, United States of America.
  • Kumar R; Oncology R & D, GlaxoSmithKline, Collegeville, Pennsylvania, United States of America.
PLoS One ; 9(6): e100880, 2014.
Article em En | MEDLINE | ID: mdl-24978597

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Neoplasias Pancreáticas / Pirazóis / Regulação Neoplásica da Expressão Gênica / Inibidores de Proteínas Quinases / Carga Tumoral / Diaminas / Antineoplásicos Idioma: En Ano de publicação: 2014 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Neoplasias Pancreáticas / Pirazóis / Regulação Neoplásica da Expressão Gênica / Inibidores de Proteínas Quinases / Carga Tumoral / Diaminas / Antineoplásicos Idioma: En Ano de publicação: 2014 Tipo de documento: Article