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Boronic Acid Transition State Inhibitors Active against KPC and Other Class A ß-Lactamases: Structure-Activity Relationships as a Guide to Inhibitor Design.
Rojas, Laura J; Taracila, Magdalena A; Papp-Wallace, Krisztina M; Bethel, Christopher R; Caselli, Emilia; Romagnoli, Chiara; Winkler, Marisa L; Spellberg, Brad; Prati, Fabio; Bonomo, Robert A.
Afiliação
  • Rojas LJ; Research Service, Louis Stokes Cleveland Department of Veterans Affairs Medical Center, Cleveland, Ohio, USA Departments of Medicine, Case Western Reserve University, Cleveland, Ohio, USA Department of Molecular Biology and Microbiology, Case Western Reserve University, Cleveland, Ohio, USA.
  • Taracila MA; Research Service, Louis Stokes Cleveland Department of Veterans Affairs Medical Center, Cleveland, Ohio, USA Departments of Medicine, Case Western Reserve University, Cleveland, Ohio, USA.
  • Papp-Wallace KM; Research Service, Louis Stokes Cleveland Department of Veterans Affairs Medical Center, Cleveland, Ohio, USA Department of Molecular Biology and Microbiology, Case Western Reserve University, Cleveland, Ohio, USA.
  • Bethel CR; Research Service, Louis Stokes Cleveland Department of Veterans Affairs Medical Center, Cleveland, Ohio, USA.
  • Caselli E; Dipartimento di Scienze della Vita, Università degli Studi di Modena e Reggio Emilia, Modena, Italy.
  • Romagnoli C; Dipartimento di Scienze della Vita, Università degli Studi di Modena e Reggio Emilia, Modena, Italy.
  • Winkler ML; Research Service, Louis Stokes Cleveland Department of Veterans Affairs Medical Center, Cleveland, Ohio, USA Departments of Medicine, Case Western Reserve University, Cleveland, Ohio, USA Department of Molecular Biology and Microbiology, Case Western Reserve University, Cleveland, Ohio, USA.
  • Spellberg B; Keck School of Medicine at University of Southern California, Los Angeles, California, USA.
  • Prati F; Dipartimento di Scienze della Vita, Università degli Studi di Modena e Reggio Emilia, Modena, Italy.
  • Bonomo RA; Research Service, Louis Stokes Cleveland Department of Veterans Affairs Medical Center, Cleveland, Ohio, USA Departments of Medicine, Case Western Reserve University, Cleveland, Ohio, USA Department of Molecular Biology and Microbiology, Case Western Reserve University, Cleveland, Ohio, USA Departme
Antimicrob Agents Chemother ; 60(3): 1751-9, 2016 Jan 04.
Article em En | MEDLINE | ID: mdl-26729496

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Triazóis / Beta-Lactamases / Ácidos Borônicos / Escherichia coli / Inibidores de beta-Lactamases / Klebsiella pneumoniae Idioma: En Ano de publicação: 2016 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Triazóis / Beta-Lactamases / Ácidos Borônicos / Escherichia coli / Inibidores de beta-Lactamases / Klebsiella pneumoniae Idioma: En Ano de publicação: 2016 Tipo de documento: Article