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Systematic development of small molecules to inhibit specific microscopic steps of Aß42 aggregation in Alzheimer's disease.
Habchi, Johnny; Chia, Sean; Limbocker, Ryan; Mannini, Benedetta; Ahn, Minkoo; Perni, Michele; Hansson, Oskar; Arosio, Paolo; Kumita, Janet R; Challa, Pavan Kumar; Cohen, Samuel I A; Linse, Sara; Dobson, Christopher M; Knowles, Tuomas P J; Vendruscolo, Michele.
Afiliação
  • Habchi J; Department of Chemistry, University of Cambridge, Cambridge CB2 1EW, United Kingdom.
  • Chia S; Department of Chemistry, University of Cambridge, Cambridge CB2 1EW, United Kingdom.
  • Limbocker R; Department of Chemistry, University of Cambridge, Cambridge CB2 1EW, United Kingdom.
  • Mannini B; Department of Chemistry, University of Cambridge, Cambridge CB2 1EW, United Kingdom.
  • Ahn M; Department of Chemistry, University of Cambridge, Cambridge CB2 1EW, United Kingdom.
  • Perni M; Department of Chemistry, University of Cambridge, Cambridge CB2 1EW, United Kingdom.
  • Hansson O; Department of Clinical Sciences, Lund University, 221 00 Lund, Sweden.
  • Arosio P; Memory Clinic, Skåne University Hospital, 205 02 Malmo, Sweden.
  • Kumita JR; Department of Chemistry, University of Cambridge, Cambridge CB2 1EW, United Kingdom.
  • Challa PK; Department of Chemistry, University of Cambridge, Cambridge CB2 1EW, United Kingdom.
  • Cohen SI; Department of Chemistry, University of Cambridge, Cambridge CB2 1EW, United Kingdom.
  • Linse S; Department of Chemistry, University of Cambridge, Cambridge CB2 1EW, United Kingdom.
  • Dobson CM; Department of Biochemistry & Structural Biology, Center for Molecular Protein Science, Lund University, 221 00 Lund, Sweden.
  • Knowles TP; Department of Chemistry, University of Cambridge, Cambridge CB2 1EW, United Kingdom; mv245@cam.ac.uk tpjk2@cam.ac.uk cmd44@cam.ac.uk.
  • Vendruscolo M; Department of Chemistry, University of Cambridge, Cambridge CB2 1EW, United Kingdom; mv245@cam.ac.uk tpjk2@cam.ac.uk cmd44@cam.ac.uk.
Proc Natl Acad Sci U S A ; 114(2): E200-E208, 2017 01 10.
Article em En | MEDLINE | ID: mdl-28011763

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Fragmentos de Peptídeos / Peptídeos beta-Amiloides / Descoberta de Drogas Limite: Animals / Humans Idioma: En Ano de publicação: 2017 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Fragmentos de Peptídeos / Peptídeos beta-Amiloides / Descoberta de Drogas Limite: Animals / Humans Idioma: En Ano de publicação: 2017 Tipo de documento: Article