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Oxazole-Bridged Combretastatin A-4 Derivatives with Tethered Hydroxamic Acids: Structure⁻Activity Relations of New Inhibitors of HDAC and/or Tubulin Function.
Schmitt, Florian; Gosch, Lisa Chiara; Dittmer, Alexandra; Rothemund, Matthias; Mueller, Thomas; Schobert, Rainer; Biersack, Bernhard; Volkamer, Andrea; Höpfner, Michael.
Afiliação
  • Schmitt F; Department of Chemistry, University of Bayreuth, Universitaetsstrasse 30, 95447 Bayreuth, Germany. florian1.schmitt@uni-bayreuth.de.
  • Gosch LC; Institute of Physiology, Charité⁻Universitätsmedizin Berlin, Charitéplatz 1, 10117 Berlin, Germany. lisa-chiara.gosch@charite.de.
  • Dittmer A; In Silico Toxicology Group, Institute of Physiology, Charité⁻Universitätsmedizin Berlin, Charitéplatz 1, 10117 Berlin, Germany. lisa-chiara.gosch@charite.de.
  • Rothemund M; Institute of Physiology, Charité⁻Universitätsmedizin Berlin, Charitéplatz 1, 10117 Berlin, Germany. alexandra.dittmer@charite.de.
  • Mueller T; Department of Chemistry, University of Bayreuth, Universitaetsstrasse 30, 95447 Bayreuth, Germany. matthias.rothemund@uni-bayreuth.de.
  • Schobert R; Internal Medicine IV, University Hospital Halle (Saale), Ernst-Grube-Str. 40, 06120 Halle, Germany. thomas.mueller@medizin.uni-halle.de.
  • Biersack B; Department of Chemistry, University of Bayreuth, Universitaetsstrasse 30, 95447 Bayreuth, Germany. rainer.schobert@uni-bayreuth.de.
  • Volkamer A; Department of Chemistry, University of Bayreuth, Universitaetsstrasse 30, 95447 Bayreuth, Germany. bernhard.biersack@yahoo.com.
  • Höpfner M; In Silico Toxicology Group, Institute of Physiology, Charité⁻Universitätsmedizin Berlin, Charitéplatz 1, 10117 Berlin, Germany. andrea.volkamer@charite.de.
Int J Mol Sci ; 20(2)2019 Jan 17.
Article em En | MEDLINE | ID: mdl-30658435

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Oxazóis / Bibenzilas / Moduladores de Tubulina / Inibidores de Histona Desacetilases / Ácidos Hidroxâmicos Tipo de estudo: Prognostic_studies Limite: Humans Idioma: En Ano de publicação: 2019 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Oxazóis / Bibenzilas / Moduladores de Tubulina / Inibidores de Histona Desacetilases / Ácidos Hidroxâmicos Tipo de estudo: Prognostic_studies Limite: Humans Idioma: En Ano de publicação: 2019 Tipo de documento: Article