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Activity of Mitragyna speciosa ("Kratom") Alkaloids at Serotonin Receptors.
León, Francisco; Obeng, Samuel; Mottinelli, Marco; Chen, Yiming; King, Tamara I; Berthold, Erin C; Kamble, Shyam H; Restrepo, Luis F; Patel, Avi; Gamez-Jimenez, Lea R; Lopera-Londoño, Carolina; Hiranita, Takato; Sharma, Abhisheak; Hampson, Aidan J; Canal, Clinton E; McMahon, Lance R; McCurdy, Christopher R.
Afiliação
  • León F; Department of Medicinal Chemistry, College of Pharmacy, University of Florida, Gainesville, Florida 32610, United States.
  • Obeng S; Department of Drug Discovery and Biomedical Sciences, College of Pharmacy, University of South Carolina, Columbia, South Carolina 29208, United States.
  • Mottinelli M; Department of Medicinal Chemistry, College of Pharmacy, University of Florida, Gainesville, Florida 32610, United States.
  • Chen Y; Department of Pharmacodynamics, College of Pharmacy, University of Florida, Gainesville, Florida 32610, United States.
  • King TI; Department of Medicinal Chemistry, College of Pharmacy, University of Florida, Gainesville, Florida 32610, United States.
  • Berthold EC; Department of Pharmaceutical Sciences, College of Pharmacy, Mercer University, Atlanta, Georgia 30341, United States.
  • Kamble SH; Department of Pharmaceutics, College of Pharmacy, University of Florida, Gainesville, Florida 32610, United States.
  • Restrepo LF; Translational Drug Development Core, Clinical and Translational Sciences Institute, University of Florida, Gainesville, Florida 32610, United States.
  • Patel A; Department of Pharmaceutics, College of Pharmacy, University of Florida, Gainesville, Florida 32610, United States.
  • Gamez-Jimenez LR; Translational Drug Development Core, Clinical and Translational Sciences Institute, University of Florida, Gainesville, Florida 32610, United States.
  • Lopera-Londoño C; Department of Pharmaceutics, College of Pharmacy, University of Florida, Gainesville, Florida 32610, United States.
  • Hiranita T; Translational Drug Development Core, Clinical and Translational Sciences Institute, University of Florida, Gainesville, Florida 32610, United States.
  • Sharma A; Department of Pharmacodynamics, College of Pharmacy, University of Florida, Gainesville, Florida 32610, United States.
  • Hampson AJ; Department of Pharmacodynamics, College of Pharmacy, University of Florida, Gainesville, Florida 32610, United States.
  • Canal CE; Department of Pharmacodynamics, College of Pharmacy, University of Florida, Gainesville, Florida 32610, United States.
  • McMahon LR; Department of Medicinal Chemistry, College of Pharmacy, University of Florida, Gainesville, Florida 32610, United States.
  • McCurdy CR; Department of Pharmacodynamics, College of Pharmacy, University of Florida, Gainesville, Florida 32610, United States.
J Med Chem ; 64(18): 13510-13523, 2021 09 23.
Article em En | MEDLINE | ID: mdl-34467758

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Receptores de Serotonina / Alcaloides de Triptamina e Secologanina / Dor Nociceptiva / Analgésicos Limite: Animals / Female / Humans / Male Idioma: En Ano de publicação: 2021 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Receptores de Serotonina / Alcaloides de Triptamina e Secologanina / Dor Nociceptiva / Analgésicos Limite: Animals / Female / Humans / Male Idioma: En Ano de publicação: 2021 Tipo de documento: Article