The ethoxycarbonyl group as both activating and protective group in <i>N</i>-acyl-Pictet-Spengler reactions using methoxystyrenes. A short approach to racemic 1-benzyltetrahydroisoquinoline alkaloids.

Keller, Marco; Sauvageot-Witzku, Karl; Geisslinger, Franz; Urban, Nicole; Schaefer, Michael; Bartel, Karin; Bracher, Franz

The ethoxycarbonyl group as both activating and protective group in N-acyl-Pictet-Spengler reactions using methoxystyrenes. A short approach to racemic 1-benzyltetrahydroisoquinoline alkaloids.

Keller, Marco; Sauvageot-Witzku, Karl; Geisslinger, Franz; Urban, Nicole; Schaefer, Michael; Bartel, Karin; Bracher, Franz.

Afiliação

Keller M; Department of Pharmacy - Center for Drug Research, Ludwig-Maximilians University, Butenandtstr. 5-13, 81377 Munich, Germany.
Sauvageot-Witzku K; Department of Pharmacy - Center for Drug Research, Ludwig-Maximilians University, Butenandtstr. 5-13, 81377 Munich, Germany.
Geisslinger F; Department of Pharmacy - Center for Drug Research, Ludwig-Maximilians University, Butenandtstr. 5-13, 81377 Munich, Germany.
Urban N; Rudolf-Boehm-Institute for Pharmacology and Toxicology, Härtelstr. 16-18, 04107 Leipzig, Germany.
Schaefer M; Rudolf-Boehm-Institute for Pharmacology and Toxicology, Härtelstr. 16-18, 04107 Leipzig, Germany.
Bartel K; Department of Pharmacy - Center for Drug Research, Ludwig-Maximilians University, Butenandtstr. 5-13, 81377 Munich, Germany.
Bracher F; Department of Pharmacy - Center for Drug Research, Ludwig-Maximilians University, Butenandtstr. 5-13, 81377 Munich, Germany.

Beilstein J Org Chem ; 17: 2716-2725, 2021.

Article em En | MEDLINE | ID: mdl-34804241