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Repurposing FDA-approved sulphonamide carbonic anhydrase inhibitors for treatment of Neisseria gonorrhoeae.
Abutaleb, Nader S; Elhassanny, Ahmed E M; Nocentini, Alessio; Hewitt, Chad S; Elkashif, Ahmed; Cooper, Bruce R; Supuran, Claudiu T; Seleem, Mohamed N; Flaherty, Daniel P.
Afiliação
  • Abutaleb NS; Department of Biomedical Sciences and Pathobiology, Virginia-Maryland College of Veterinary Medicine, Virginia Polytechnic Institute and State University, Blacksburg, VI, USA.
  • Elhassanny AEM; Department of Biomedical Sciences and Pathobiology, Virginia-Maryland College of Veterinary Medicine, Virginia Polytechnic Institute and State University, Blacksburg, VI, USA.
  • Nocentini A; Department of NEUROFARBA, Section of Pharmaceutical and Nutraceutical Sciences, University of Florence, Polo Scientifico, Firenze, Italy.
  • Hewitt CS; Department of Medicinal Chemistry and Molecular Pharmacology, College of Pharmacy, Purdue University, West Lafayette, IN, USA.
  • Elkashif A; Department of Comparative Pathobiology, College of Veterinary Medicine, Purdue University, West Lafayette, IN, USA.
  • Cooper BR; Metabolite Profiling Facility, Bindley Bioscience Center, Purdue University, West Lafayette, Indiana, United States.
  • Supuran CT; Department of NEUROFARBA, Section of Pharmaceutical and Nutraceutical Sciences, University of Florence, Polo Scientifico, Firenze, Italy.
  • Seleem MN; Department of Biomedical Sciences and Pathobiology, Virginia-Maryland College of Veterinary Medicine, Virginia Polytechnic Institute and State University, Blacksburg, VI, USA.
  • Flaherty DP; Center for Emerging, Zoonotic and Arthropod-borne Pathogens, Virginia Polytechnic Institute and State University, Blacksburg, VI, USA.
J Enzyme Inhib Med Chem ; 37(1): 51-61, 2022 Dec.
Article em En | MEDLINE | ID: mdl-34894972

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Inibidores da Anidrase Carbônica / Anidrases Carbônicas / Etoxzolamida / Acetazolamida / Antibacterianos / Neisseria gonorrhoeae Tipo de estudo: Risk_factors_studies País/Região como assunto: America do norte Idioma: En Ano de publicação: 2022 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Inibidores da Anidrase Carbônica / Anidrases Carbônicas / Etoxzolamida / Acetazolamida / Antibacterianos / Neisseria gonorrhoeae Tipo de estudo: Risk_factors_studies País/Região como assunto: America do norte Idioma: En Ano de publicação: 2022 Tipo de documento: Article