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Design and biological evaluation of substituted 5,7-dihydro-6H-indolo[2,3-c]quinolin-6-one as novel selective Haspin inhibitors.
Avula, Sreenivas; Peng, Xudan; Lang, Xingfen; Tortorella, Micky; Josselin, Béatrice; Bach, Stéphane; Bourg, Stephane; Bonnet, Pascal; Buron, Frédéric; Ruchaud, Sandrine; Routier, Sylvain; Neagoie, Cleopatra.
Afiliação
  • Avula S; Guangzhou Institute of Biomedicine and Health, Chinese Academy of Science, Guangzhou, China.
  • Peng X; Guangzhou Institute of Biomedicine and Health, Chinese Academy of Science, Guangzhou, China.
  • Lang X; Guangzhou Institute of Biomedicine and Health, Chinese Academy of Science, Guangzhou, China.
  • Tortorella M; Guangzhou Institute of Biomedicine and Health, Chinese Academy of Science, Guangzhou, China.
  • Josselin B; Centre for Regenerative Medicine and Health, Hong Kong Institute of Science and Innovation, Chinese Academy of Science, Hong Kong SAR, China.
  • Bach S; Sorbonne Université/CNRS UMR8227, Roscoff cedex, France.
  • Bourg S; Sorbonne Université/CNRS FR2424, Plateforme de criblage KISSf (Kinase Inhibitor Specialized Screening Facility), Roscoff cedex, France.
  • Bonnet P; Sorbonne Université/CNRS UMR8227, Roscoff cedex, France.
  • Buron F; Sorbonne Université/CNRS FR2424, Plateforme de criblage KISSf (Kinase Inhibitor Specialized Screening Facility), Roscoff cedex, France.
  • Ruchaud S; Institut de Chimie Organique et Analytique, Université d'Orléans, UMR CNRS 7311, Orleans, France.
  • Routier S; Institut de Chimie Organique et Analytique, Université d'Orléans, UMR CNRS 7311, Orleans, France.
  • Neagoie C; Institut de Chimie Organique et Analytique, Université d'Orléans, UMR CNRS 7311, Orleans, France.
J Enzyme Inhib Med Chem ; 37(1): 1632-1650, 2022 Dec.
Article em En | MEDLINE | ID: mdl-35670091

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Neoplasias Ósseas / Quinolonas Limite: Humans Idioma: En Ano de publicação: 2022 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Neoplasias Ósseas / Quinolonas Limite: Humans Idioma: En Ano de publicação: 2022 Tipo de documento: Article