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Synthesis and biological activity evaluation of 3-(hetero) arylideneindolin-2-ones as potential c-Src inhibitors.
Princiotto, Salvatore; Musso, Loana; Manetti, Fabrizio; Marcellini, Valentina; Maga, Giovanni; Crespan, Emmanuele; Perini, Cecilia; Zaffaroni, Nadia; Beretta, Giovanni Luca; Dallavalle, Sabrina.
Afiliação
  • Princiotto S; Department of Food, Environmental and Nutritional Sciences (DeFENS), University of Milan, Milan, Italy.
  • Musso L; Department of Food, Environmental and Nutritional Sciences (DeFENS), University of Milan, Milan, Italy.
  • Manetti F; Dipartimento di Biotecnologie, Chimica e Farmacia, Università di Siena, Siena, Italy.
  • Marcellini V; Dipartimento di Biotecnologie, Chimica e Farmacia, Università di Siena, Siena, Italy.
  • Maga G; Institute of Molecular Genetics IGM, CNR "Luigi Luca Cavalli-Sforza", Pavia, Italy.
  • Crespan E; Institute of Molecular Genetics IGM, CNR "Luigi Luca Cavalli-Sforza", Pavia, Italy.
  • Perini C; Institute of Molecular Genetics IGM, CNR "Luigi Luca Cavalli-Sforza", Pavia, Italy.
  • Zaffaroni N; Molecular Pharmacology Unit, Department of Applied Research and Technological Development, Fondazione IRCCS Istituto Nazionale Tumori, Milan, Italy.
  • Beretta GL; Molecular Pharmacology Unit, Department of Applied Research and Technological Development, Fondazione IRCCS Istituto Nazionale Tumori, Milan, Italy.
  • Dallavalle S; Department of Food, Environmental and Nutritional Sciences (DeFENS), University of Milan, Milan, Italy.
J Enzyme Inhib Med Chem ; 37(1): 2382-2394, 2022 Dec.
Article em En | MEDLINE | ID: mdl-36050846

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Inibidores de Proteínas Quinases / Antineoplásicos Idioma: En Ano de publicação: 2022 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Inibidores de Proteínas Quinases / Antineoplásicos Idioma: En Ano de publicação: 2022 Tipo de documento: Article