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Discovery of selective and potent USP22 inhibitors via structure-based virtual screening and bioassays exerting anti-tumor activity.
Zhang, Yue; Song, Jiankun; Zhou, Yuanzhang; Jia, Huijun; Zhou, Tianyu; Sun, Yingbo; Gao, Qiong; Zhao, Yue; Pan, Yujie; Sun, Zhaolin; Chu, Peng.
Afiliação
  • Zhang Y; College of Pharmacy, Dalian Medical University, Dalian 116044, China.
  • Song J; Department of Biochemistry and Molecular Biology, Dalian Medical University, Dalian 116044, China.
  • Zhou Y; Department of Biochemistry and Molecular Biology, Dalian Medical University, Dalian 116044, China.
  • Jia H; Department of Biochemistry and Molecular Biology, Dalian Medical University, Dalian 116044, China.
  • Zhou T; College of Pharmacy, Dalian Medical University, Dalian 116044, China.
  • Sun Y; College of Pharmacy, Dalian Medical University, Dalian 116044, China.
  • Gao Q; Department of Biochemistry and Molecular Biology, Dalian Medical University, Dalian 116044, China.
  • Zhao Y; Department of Biochemistry and Molecular Biology, Dalian Medical University, Dalian 116044, China.
  • Pan Y; College of Pharmacy, Dalian Medical University, Dalian 116044, China.
  • Sun Z; College of Pharmacy, Dalian Medical University, Dalian 116044, China; Department of Biochemistry and Molecular Biology, Dalian Medical University, Dalian 116044, China. Electronic address: zlsun56@yeah.net.
  • Chu P; College of Pharmacy, Dalian Medical University, Dalian 116044, China. Electronic address: chupeng0801@163.com.
Bioorg Chem ; 141: 106842, 2023 12.
Article em En | MEDLINE | ID: mdl-37769523

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Sirtuína 1 / Antígeno B7-H1 Tipo de estudo: Diagnostic_studies / Screening_studies Limite: Humans Idioma: En Ano de publicação: 2023 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Sirtuína 1 / Antígeno B7-H1 Tipo de estudo: Diagnostic_studies / Screening_studies Limite: Humans Idioma: En Ano de publicação: 2023 Tipo de documento: Article