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Superiority of the Triple-Acting 5-HT6R/5-HT3R Antagonist and MAO-B Reversible Inhibitor PZ-1922 over 5-HT6R Antagonist Intepirdine in Alleviation of Cognitive Deficits in Rats.
Grychowska, Katarzyna; López-Sánchez, Uriel; Vitalis, Mathieu; Canet, Geoffrey; Satala, Grzegorz; Olejarz-Maciej, Agnieszka; Golebiowska, Joanna; Kurczab, Rafal; Pietrus, Wojciech; Kubacka, Monika; Moreau, Christophe; Walczak, Maria; Blicharz-Futera, Klaudia; Bento, Ophélie; Bantreil, Xavier; Subra, Gilles; Bojarski, Andrzej J; Lamaty, Frédéric; Becamel, Carine; Zussy, Charleine; Chaumont-Dubel, Séverine; Popik, Piotr; Nury, Hugues; Marin, Philippe; Givalois, Laurent; Zajdel, Pawel.
Afiliação
  • Grychowska K; Faculty of Pharmacy, Jagiellonian University Medical College, 9 Medyczna Str., 30-688 Kraków, Poland.
  • López-Sánchez U; Univ. Grenoble Alpes, CNRS, CEA, IBS, F-38000 Grenoble, France.
  • Vitalis M; Molecular Mechanisms in Neurodegenerative Dementia (MMDN) Laboratory, University of Montpellier, EPHE-PSL, INSERM U1198, 34-095 Montpellier, France.
  • Canet G; Faculty of Medicine, Laval University, CR-CHUQ, G1 V 4G2 Québec City (QC), Canada.
  • Satala G; Maj Institute of Pharmacology, Polish Academy of Sciences, 12 Smetna Str., 31-324 Kraków, Poland.
  • Olejarz-Maciej A; Faculty of Pharmacy, Jagiellonian University Medical College, 9 Medyczna Str., 30-688 Kraków, Poland.
  • Golebiowska J; Maj Institute of Pharmacology, Polish Academy of Sciences, 12 Smetna Str., 31-324 Kraków, Poland.
  • Kurczab R; Maj Institute of Pharmacology, Polish Academy of Sciences, 12 Smetna Str., 31-324 Kraków, Poland.
  • Pietrus W; Maj Institute of Pharmacology, Polish Academy of Sciences, 12 Smetna Str., 31-324 Kraków, Poland.
  • Kubacka M; Faculty of Pharmacy, Jagiellonian University Medical College, 9 Medyczna Str., 30-688 Kraków, Poland.
  • Moreau C; Univ. Grenoble Alpes, CNRS, CEA, IBS, F-38000 Grenoble, France.
  • Walczak M; Faculty of Pharmacy, Jagiellonian University Medical College, 9 Medyczna Str., 30-688 Kraków, Poland.
  • Blicharz-Futera K; Faculty of Pharmacy, Jagiellonian University Medical College, 9 Medyczna Str., 30-688 Kraków, Poland.
  • Bento O; IBMM, Université de Montpellier, CNRS, ENSCM, 34-293 Montpellier, France.
  • Bantreil X; Institut de Génomique Fonctionnelle, Université de Montpellier, CNRS, INSERM, 34-094 Montpellier, France.
  • Subra G; IBMM, Université de Montpellier, CNRS, ENSCM, 34-293 Montpellier, France.
  • Bojarski AJ; IBMM, Université de Montpellier, CNRS, ENSCM, 34-293 Montpellier, France.
  • Lamaty F; Maj Institute of Pharmacology, Polish Academy of Sciences, 12 Smetna Str., 31-324 Kraków, Poland.
  • Becamel C; IBMM, Université de Montpellier, CNRS, ENSCM, 34-293 Montpellier, France.
  • Zussy C; Institut de Génomique Fonctionnelle, Université de Montpellier, CNRS, INSERM, 34-094 Montpellier, France.
  • Chaumont-Dubel S; Molecular Mechanisms in Neurodegenerative Dementia (MMDN) Laboratory, University of Montpellier, EPHE-PSL, INSERM U1198, 34-095 Montpellier, France.
  • Popik P; Institut de Génomique Fonctionnelle, Université de Montpellier, CNRS, INSERM, 34-094 Montpellier, France.
  • Nury H; Maj Institute of Pharmacology, Polish Academy of Sciences, 12 Smetna Str., 31-324 Kraków, Poland.
  • Marin P; Univ. Grenoble Alpes, CNRS, CEA, IBS, F-38000 Grenoble, France.
  • Givalois L; Institut de Génomique Fonctionnelle, Université de Montpellier, CNRS, INSERM, 34-094 Montpellier, France.
  • Zajdel P; Molecular Mechanisms in Neurodegenerative Dementia (MMDN) Laboratory, University of Montpellier, EPHE-PSL, INSERM U1198, 34-095 Montpellier, France.
J Med Chem ; 66(21): 14928-14947, 2023 11 09.
Article em En | MEDLINE | ID: mdl-37797083

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Serotonina / Doença de Alzheimer Tipo de estudo: Prognostic_studies Limite: Animals Idioma: En Ano de publicação: 2023 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Assunto principal: Serotonina / Doença de Alzheimer Tipo de estudo: Prognostic_studies Limite: Animals Idioma: En Ano de publicação: 2023 Tipo de documento: Article