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Investigation of novel bis-thiadiazole bearing schiff base derivatives as effective inhibitors of thymidine phosphorylase: Synthesis, in vitro bioactivity and molecular docking study.
Hussain, Rafaqat; Rehman, Wajid; Khan, Shoaib; Jaber, Fadi; Rahim, Fazal; Shah, Mazloom; Khan, Yousaf; Iqbal, Shahid; Naz, Haseena; Khan, Imran; Issa Alahmdi, Mohammed; Awwad, Nasser S; Ibrahium, Hala A.
Afiliação
  • Hussain R; Department of Chemistry, Hazara University, Mansehra 21120, Pakistan.
  • Rehman W; Department of Chemistry, Hazara University, Mansehra 21120, Pakistan.
  • Khan S; Department of Chemistry, Abbottabad University of Science and Technology (AUST), Abbottabad, Pakistan.
  • Jaber F; Department of Biomedical Engineering, Ajman University, Ajman, United Arab Emirates.
  • Rahim F; Center of Medical and Bio-Allied Health Sciences Research, Ajman University, Ajman, United Arab Emirates.
  • Shah M; Department of Chemistry, Hazara University, Mansehra 21120, Pakistan.
  • Khan Y; Department of Chemistry, Faculty of Science, Grand Asian University, Sialkot, Pakistan.
  • Iqbal S; Department of Chemistry, COMSATS University, Islamabad 45550, Pakistan.
  • Naz H; Nottingham Ningbo China Beacons of Excellence Research and Innovation Institute, University of Nottingham, Ningbo 315100, China.
  • Khan I; Department of Chemistry, Hazara University, Mansehra 21120, Pakistan.
  • Issa Alahmdi M; Department of Chemistry, Hazara University, Mansehra 21120, Pakistan.
  • Awwad NS; Department of Chemistry, Faculty of Science, University of Tabuk, Tabuk 71491, Saudi Arabia.
  • Ibrahium HA; Chemistry Department, Faculty of Science, King Khalid University, P.O. Box 9004, Abha 61413, Saudi Arabia.
Saudi Pharm J ; 31(11): 101823, 2023 Nov.
Article em En | MEDLINE | ID: mdl-37965293

Texto completo: 1 Base de dados: MEDLINE Idioma: En Ano de publicação: 2023 Tipo de documento: Article

Texto completo: 1 Base de dados: MEDLINE Idioma: En Ano de publicação: 2023 Tipo de documento: Article