Search details
1.
Design and development of a series of borocycles as selective, covalent kallikrein 5 inhibitors.
Bioorg Med Chem Lett
; 29(20): 126675, 2019 10 15.
Article
in English
| MEDLINE | ID: mdl-31521475
2.
The discovery of potent and selective kynurenine 3-monooxygenase inhibitors for the treatment of acute pancreatitis.
Bioorg Med Chem Lett
; 27(9): 2023-2028, 2017 05 01.
Article
in English
| MEDLINE | ID: mdl-28336141
3.
Corrigendum to 'Design and development of a series of borocycles as selective, covalent kallikrein 5 inhibitors' [Bioorg. Med. Chem. Lett. 29 (2019) 126675].
Bioorg Med Chem Lett
; 30(2): 126771, 2020 Jan 15.
Article
in English
| MEDLINE | ID: mdl-31859161
4.
From ApoA1 upregulation to BET family bromodomain inhibition: discovery of I-BET151.
Bioorg Med Chem Lett
; 22(8): 2963-7, 2012 Apr 15.
Article
in English
| MEDLINE | ID: mdl-22386529
5.
Identification of a novel series of BET family bromodomain inhibitors: binding mode and profile of I-BET151 (GSK1210151A).
Bioorg Med Chem Lett
; 22(8): 2968-72, 2012 Apr 15.
Article
in English
| MEDLINE | ID: mdl-22437115
6.
A Potent and Selective Kallikrein-5 Inhibitor Delivers High Pharmacological Activity in Skin from Patients with Netherton Syndrome.
J Invest Dermatol
; 141(9): 2272-2279, 2021 09.
Article
in English
| MEDLINE | ID: mdl-33744298
7.
Design and evaluation of a novel series of 2,3-oxidosqualene cyclase inhibitors with low systemic exposure, relationship between pharmacokinetic properties and ocular toxicity.
Bioorg Med Chem
; 16(11): 6218-32, 2008 Jun 01.
Article
in English
| MEDLINE | ID: mdl-18467104
8.
Development of a Series of Kynurenine 3-Monooxygenase Inhibitors Leading to a Clinical Candidate for the Treatment of Acute Pancreatitis.
J Med Chem
; 60(8): 3383-3404, 2017 04 27.
Article
in English
| MEDLINE | ID: mdl-28398044
9.
Naphthyridines as novel BET family bromodomain inhibitors.
ChemMedChem
; 9(3): 580-9, 2014 Mar.
Article
in English
| MEDLINE | ID: mdl-24000170
10.
Comparison of soluble guanylate cyclase stimulators and activators in models of cardiovascular disease associated with oxidative stress.
Front Pharmacol
; 3: 128, 2012.
Article
in English
| MEDLINE | ID: mdl-22783192
11.
Discovery and characterization of small molecule inhibitors of the BET family bromodomains.
J Med Chem
; 54(11): 3827-38, 2011 Jun 09.
Article
in English
| MEDLINE | ID: mdl-21568322
12.
Pharmacological inhibition of stearoyl-CoA desaturase 1 improves insulin sensitivity in insulin-resistant rat models.
Eur J Pharmacol
; 618(1-3): 28-36, 2009 Sep 15.
Article
in English
| MEDLINE | ID: mdl-19616540
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